Search Count: 21
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Human Prmt5:Mep50 Complex In Complex With Ligand 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-09-10 Classification: TRANSLOCASE Ligands: A1CHO, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1CHO, EDO, GOL
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Co-Crystal Structure Of Krit1 With A 1-Hydroxy 2-Naphthaldehyde Derivative (6-Ethynyl-2-Hydroxy-1-Naphthaldehyde)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2023-12-13 Classification: CELL ADHESION Ligands: XHZ, MG, GNP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-13
Ligands: XHZ, MG, GNP
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Co-Crystal Structure Of Krit1 With A 1-Hydroxy 2-Naphthaldehyde Derivative (6-(Furan-2-Yl)-2-Hydroxy-1-Naphthaldehyde).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2023-12-06 Classification: CELL ADHESION Ligands: XE2, MG, GNP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: XE2, MG, GNP
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Co-Crystal Structure Of Krit1 With A 1-Hydroxy 2-Naphthaldehyde Derivative (6-(Furan-2-Yl)-2-Hydroxy-1-Naphthaldehyde)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2023-12-06 Classification: CELL ADHESION Ligands: ZTA, MG, GNP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: ZTA, MG, GNP
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Fragment-Based Discovery Of A Novel Bruton'S Tyrosine Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: IMD, PGO, 0BQ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: IMD, PGO, 0BQ, EDO
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Fragment-Based Discovery Of A Novel Bruton'S Tyrosine Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: IMD, EDO, DMS, 0UW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: IMD, EDO, DMS, 0UW
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Fragment-Based Discovery Of A Novel Bruton'S Tyrosine Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: IMD, PGO, DMS, 0GW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: IMD, PGO, DMS, 0GW
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Fragment-Based Drug Design Of A Novel, Covalent Bruton'S Tyrosine Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: IMD, 0CI, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: IMD, 0CI, DMS
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Met Tyrosine Kinase Inhibition Enhances The Antitumor Efficacy Of An Hgf Antibody
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-02-12 Classification: TRANSFERASE-TRANSFERASE INHIBITOR Ligands: 84S, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-12
Ligands: 84S, CL
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Met Tyrosine Kinase Inhibition Enhances The Antitumor Efficacy Of An Hgf Antibody
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-05-31 Classification: TRANSFERASE/INHIBITOR Ligands: 84M, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: 84M, GOL, CL
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Met Tyrosine Kinase Inhibition Enhances The Antitumor Efficacy Of An Hgf Antibody
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2017-05-31 Classification: TRANSFERASE/INHIBITOR Ligands: 84P, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: 84P, CL
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Alk-5 Kinase Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2017-04-12 Classification: Transferase/Transferase Inhibitor Ligands: 8LY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-12
Ligands: 8LY
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Crystal Structure Of Autotaxin/Enpp2 With A Covalent Fragment
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2017-03-15 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, NAG, ACT, 6C1 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: ZN, CA, NAG, ACT, 6C1
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Crystal Structure Of Mouse Comt Bound To An Inhibitor
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2014-06-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2F6 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2014-06-25
Ligands: 2F6
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Parp Complexed With Benzo[1,4]Oxazin-3-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-08-07 Classification: transferase/transferase inhibitor Ligands: 1WQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-07
Ligands: 1WQ
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Crystal Structure Of The Vegfr2 Kinase Domain In Complex With A Back Pocket Binder
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2012-09-05 Classification: TRANSFERASE Ligands: BPK, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-05
Ligands: BPK, EDO
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Crystal Structure Of Human Vegfr2 Kinase Domain With Compound A.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2012-08-15 Classification: TRANSFERASE Ligands: 4TT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-15
Ligands: 4TT
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Clostridium Botulinum Serotype A Light Chain Inhibited By 4-Chlorocinnamic Hydroxamate
Organism: Clostridium botulinum
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2007-06-05 Classification: HYDROLASE Ligands: ZN, PO4, GB5 |
Organism: Clostridium botulinum
Method: X-RAY DIFFRACTION
Release Date: 2007-06-05
Ligands: ZN, PO4, GB5
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Clostridium Botulinum Neurotoxin Serotype A Light Chain Inhibited By 2,4-Dichlorocinnamic Hydroxamate
Organism: Clostridium botulinum
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2007-06-05 Classification: HYDROLASE Ligands: ZN, GB4 |
Organism: Clostridium botulinum
Method: X-RAY DIFFRACTION
Release Date: 2007-06-05
Ligands: ZN, GB4
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Clostridium Botulinum Neurotoxin Serotype A Light Chain Inhibited By L-Arginine Hydroxamate
Organism: Clostridium botulinum
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2007-06-05 Classification: HYDROLASE Ligands: ZN, AHL |
Organism: Clostridium botulinum
Method: X-RAY DIFFRACTION
Release Date: 2007-06-05
Ligands: ZN, AHL
