Search Count: 18
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Estrogen Receptor Alpha Ligand Binding Domain In Complex With Palazestrant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-03-19 Classification: TRANSCRIPTION Ligands: A1AEA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-19
Ligands: A1AEA, GOL
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Usp7 In Complex With Gne6640 (4-(2-Amino-4-Ethyl-5-(1H-Indazol-5-Yl)Pyridin-3-Yl)Phenol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2017-10-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 8JM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-25
Ligands: 8JM
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Usp7 In Complex With Gne6776 (6'-Amino-4'-Ethyl-5'-(4-Hydroxyphenyl)-N-Methyl-[3,3'-Bipyridine]-6-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2017-10-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 8JP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-25
Ligands: 8JP
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Crystal Structure Of The Apo-Form Of Usp7 Catalytic Domain [V302K] Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-08-09 Classification: HYDROLASE Ligands: GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
Ligands: GOL
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Crystal Structure Of Usp7 Catalytic Domain [V302K] Mutant In Complex With Ubiquitin (Malonate Bound)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2017-08-09 Classification: HYDROLASE Ligands: MLA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
Ligands: MLA, GOL
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Crystal Structure Of Usp7 Catalytic Domain [V302K] Mutant In Complex With Ubiquitin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2017-08-09 Classification: HYDROLASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
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Crystal Structure Of Usp7 Catalytic Domain [H294E] Mutant In Complex With Ubiquitin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2017-08-09 Classification: HYDROLASE Ligands: EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
Ligands: EPE
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Crystal Structure Of Usp7 Catalytic Domain [L299A] Mutant In Complex With Ubiquitin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2017-08-09 Classification: HYDROLASE Ligands: GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
Ligands: GOL
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Crystal Structure Of Kaposi'S Sarcoma-Associated Herpesvirus (Kshv) Protease In Complex With Dimer Disruptor
Organism: Human herpesvirus 8
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2014-07-23 Classification: HYDROLASE Ligands: 25G, GOL, DMS |
Organism: Human herpesvirus 8
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: 25G, GOL, DMS
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Crystal Structure Of Kaposi'S Sarcoma-Associated Herpesvirus (Kshv) Protease In Complex With A Dimer Disruptor
Organism: Human herpesvirus 8
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2014-07-16 Classification: HYDROLASE Ligands: 24Q, DMS |
Organism: Human herpesvirus 8
Method: X-RAY DIFFRACTION
Release Date: 2014-07-16
Ligands: 24Q, DMS
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Tailoring Small Molecules For An Allosteric Site On Procaspase-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2014-01-01 Classification: hydrolase/hydrolase inhibitor Ligands: PO4, 2GQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-01
Ligands: PO4, 2GQ
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Tailoring Small Molecules For An Allosteric Site On Procaspase-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2014-01-01 Classification: hydrolase/hydrolase inhibitor Ligands: 2J5, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-01
Ligands: 2J5, PO4
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Tailoring Small Molecules For An Allosteric Site On Procaspase-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2014-01-01 Classification: hydrolase/hydrolase inhibitor Ligands: 2J6, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-01
Ligands: 2J6, PO4
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Tailoring Small Molecules For An Allosteric Site On Procaspase-6: Cpd1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2013-12-18 Classification: hydrolase/hydrolase inhibitor Ligands: 2FQ, PO4, MPD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-18
Ligands: 2FQ, PO4, MPD
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Tailoring Small Molecules For An Allosteric Site On Procaspase-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2013-12-18 Classification: hydrolase/hydrolase inhibitor Ligands: PO4, 2GQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-18
Ligands: PO4, 2GQ
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Tailoring Small Molecules For An Allosteric Site On Procaspase-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2013-12-18 Classification: HYDROLASE Ligands: 2GQ, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-18
Ligands: 2GQ, PO4
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Tailoring Small Molecules For An Allosteric Site On Procaspase-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2013-12-18 Classification: hydrolase/hydrolase inhibitor Ligands: PO4, 2J7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-18
Ligands: PO4, 2J7
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Mechanistic And Structural Understanding Of Uncompetitive Inhibitors Of Caspase-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2013-03-20 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 4HV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: 4HV
