Structural Entry Filters:

Search Count: 26

Download
6VIW image
Brd4_Bromodomain1 Complex With Pyrrolopyridone Compound 18

6VIX image
Brd4_Bromodomain2 Complex With Pyrrolopyridone Compound 18

6VIY image
Brd2_Bromodomain2 Complex With Pyrrolopyridone Compound 27

6VIZ image
Brd4_Bromodomain1 Complex With Pyrrolopyridone Compound 27

6ONY image
Brd2_Bromodomain1 Complex With Inhibitor 744

6E6J image
Brd2_Bromodomain2 Complex With Inhibitor 744

6B4L image
Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor

6B4U image
Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor



5UEW image
Brd2 Bromodomain2 With A-1360579




5VKC image
Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor

4QVX image
Discovery Of A Potent And Selective Bcl-Xl Inhibitor That Demonstrates Thrombocytopenia And Inhibits Tumor Growth In Vivo

4TUH image
Bcl-Xl In Complex With Inhibitor (Compound 10)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2014-10-15
Classification: APOPTOSIS
Ligands: 38H, EDO, ACT

3JXW image
Discovery Of 3H-Benzo[4,5]Thieno[3,2-D]Pyrimidin-4-Ones As Potent, Highly Selective And Orally Bioavailable Pim Kinases Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2009-11-10
Classification: TRANSFERASE
Ligands: LXG

3JY0 image
Discovery Of 3H-Benzo[4,5]Thieno[3,2-D]Pyrimidin-4-Ones As Potent, Highly Selective And Orally Bioavailable Pim Kinases Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2009-11-10
Classification: TRANSFERASE
Ligands: LYG

3JYA image
Discovery Of 3H-Benzo[4,5]Thieno[3,2-D]Pyrimidin-4-Ones As Potent, Highly Selective And Orally Bioavailable Pim Kinases Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2009-11-10
Classification: TRANSFERASE
Ligands: LWG
Protein Functional Filters:
Feedback Form
Name
Email
Institute
Feedback