Search Count: 121
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Discovery Of An Orally Biovailable Kras G12D Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.36 Å Release Date: 2025-01-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GDP, MG, A1BEI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: GDP, MG, A1BEI
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Discovery Of An Orally Bioavailable Kras G12D Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2025-01-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GDP, A1BEJ, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: GDP, A1BEJ, MG
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Tead2 With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2023-12-13 Classification: SIGNALING PROTEIN Ligands: MYR, B3F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-13
Ligands: MYR, B3F
 |
Tead2 With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-12-13 Classification: SIGNALING PROTEIN Ligands: F3Y, MYR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-13
Ligands: F3Y, MYR
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Tead2 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN Ligands: MYR, GOL, WJC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: MYR, GOL, WJC
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Tead2 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN Ligands: MYR, ZUL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: MYR, ZUL
 |
Tead2 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN Ligands: ZUP, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: ZUP, GOL
 |
Tead2 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN Ligands: MYR, ZUT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: MYR, ZUT
 |
Histone-Lysine N-Methyltransferase Nsd2-Pwwp1 With Compound Mrt10241866A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2021-05-05 Classification: TRANSFERASE Ligands: Y6V, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: Y6V, UNX
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Histone-Lysine N-Methyltransferase Nsd2-Pwwp1 With Compound Unc6934
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: V01, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: V01, UNX
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Pwwp1 Domain Of Nsd2 In Complex With Mr837
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-11-13 Classification: TRANSFERASE Ligands: Q5D, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-13
Ligands: Q5D, UNX
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EH2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EH2
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHQ
 |
X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHE
 |
X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHK
 |
X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EH8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EH8
 |
X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHT
 |
X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHH
 |
X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHW
 |
X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound Bi-9321
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EJE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EJE