Search Count: 17
 |
Smarca2 Bromodomain In Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2025-01-15 Classification: GENE REGULATION Ligands: ZN, A1A1O, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: ZN, A1A1O, EDO, ACT
 |
Smarca2 Bromodomain In Complex With Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2025-01-15 Classification: GENE REGULATION Ligands: ZN, A1A1P, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: ZN, A1A1P, ACT
 |
Discovery Of Potent, Highly Selective And Efficacious Smarca2 Degraders - Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: A1BF5, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1BF5, ZN
 |
Discovery Of Potent, Highly Selective And Efficacious Smarca2 Degraders - Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: A1A1O, ZN, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1O, ZN, ACT
 |
Discovery Of Potent, Highly Selective And Efficacious Smarca2 Degraders - Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: A1A1P, ZN, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1P, ZN, ACT
 |
Crystal Structure Of The Human Brd2 Bd1 Bromodomain In Complex With 9-(Cyclopropylmethyl)-7-[(2R,6S)-2,6-Dimethylmorpholine-4-Carbonyl]-3-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-9H-Carbazole-1-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YW1, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YW1, EDO
 |
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With 9-Benzyl-2-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-7-(2-Hydroxypropan-2-Yl)-9H-Carbazole-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YW4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YW4, EDO
 |
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With 2-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-7-(2-Hydroxypropan-2-Yl)-9-[(S)-(Oxan-4-Yl)(Phenyl)Methyl]-9H-Carbazole-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YW7, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YW7, EDO
 |
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Bms-986158, 2-{3-(1,4-Dimethyl-1H-1,2,3-Triazol-5-Yl)-5-[(S)-(Oxan-4-Yl)(Phenyl)Methyl]-5H-Pyrido[3,2-B]Indol-7-Yl}Propan-2-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YWA, IOD, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YWA, IOD, EDO
 |
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7G
 |
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7H
 |
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7I
 |
Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2020-06-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Z7F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-17
Ligands: Z7F
 |
Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-04-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TKJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: TKJ
 |
Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2020-04-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Z7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: Z7D
 |
Tgf-Beta Receptor Type 1 Kinase Domain (T204D) In Complex With N-(3-Fluoropyridin-4-Yl)-2-[6-(Trifluoromethyl)Pyridin-2-Yl]-7H-Pyrrolo[2,3-D]Pyrimidin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2018-02-07 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: D0A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-07
Ligands: D0A
 |
Structure Of Janus Kinase 2 With A Pyrrolotriazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-02-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J2I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-16
Ligands: J2I