Search Count: 13
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O67 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O67
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O5V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O5V
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, O5Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: MG, GDP, O5Y
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O5S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O5S
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Crystal Structure Of An Extender (Spd28345)-Modified Human Pdk1 Complex 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2011-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SYP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-20
Ligands: SYP
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Pdk1 In Complex With Dfg-Out Inhibitor Xxx
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MP7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-20
Ligands: MP7
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Crystal Structure Of The Mouse Aurora-A Catalytic Domain (Asn186->Gly, Lys240->Arg, Met302->Leu) In Complex With Compound 290.
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2009-05-05 Classification: TRANSFERASE Ligands: AK5 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2009-05-05
Ligands: AK5
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Crystal Structure Of The Mouse Aurora-A Catalytic Domain (Asn186->Gly, Lys240->Arg, Met302->Leu) In Complex With Compound 823.
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2009-05-05 Classification: TRANSFERASE Ligands: AK6 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2009-05-05
Ligands: AK6
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Crystal Structure Of The Mouse Aurora-A Catalytic Domain (Asn186->Gly, Lys240->Arg, Met302->Leu) In Complex With Compound 130.
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2009-05-05 Classification: TRANSFERASE Ligands: AK7 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2009-05-05
Ligands: AK7
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Allosteric Inhibition Of Protein Tyrosine Phosphatase 1B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2004-07-20 Classification: HYDROLASE Ligands: BB3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-07-20
Ligands: BB3
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Allosteric Inhibition Of Protein Tyrosine Phosphatase 1B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2004-07-20 Classification: HYDROLASE Ligands: MG, 892 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-07-20
Ligands: MG, 892
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Allosteric Inhibition Of Protein Tyrosine Phosphatase 1B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2004-07-20 Classification: HYDROLASE Ligands: FRJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-07-20
Ligands: FRJ
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Ptp1B R47C Modified At C47 With N-[4-(2-{2-[3-(2-Bromo-Acetylamino)-Propionylamino]-3-Hydroxy-Propionylamino}-Ethyl)-Phenyl]-Oxalamic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2003-05-06 Classification: HYDROLASE Ligands: FG1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-05-06
Ligands: FG1
