Search Count: 9
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Highly Potent And Selective 3-N-Methylquinazoline-4(3H)-One Based Inhibitors Of B-Rafv600E Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2014-04-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2VX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-09
Ligands: 2VX
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B-Raf Kinase Domain In Complex With An Aminothienopyrimidine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2013-04-24 Classification: Transferase/Transferase Inhibitor Ligands: RI8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: RI8
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B-Raf Kinase Domain In Complex With An Aminopyridimine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2013-04-24 Classification: Transferase/Transferase Inhibitor Ligands: RI9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: RI9
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Crystal Structure Of B-Raf Kinase Domain In Complex With A Dihydropyrido[2,3-D]Pyrimidinone-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2012-05-09 Classification: Transferase/Transferase Inhibitor Ligands: T1Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-09
Ligands: T1Q
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Human B-Raf Kinase Domain In Complex With An Bromopyridine Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2011-10-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TV4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: TV4
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Human B-Raf Kinase Domain In Complex With A Methoxypyrazolopyridinyl Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2011-10-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B0R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: B0R
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Human B-Raf Kinase In Complex With An Amide Linked Pyrazolopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2011-08-17 Classification: Transferase/Transferase Inhibitor Ligands: BR2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-17
Ligands: BR2
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Non-Oxime Pyrazole Based Inhibitors Of B-Raf Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2011-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SM7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-18
Ligands: SM7
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Pyrazole-Based Inhibitors Of B-Raf Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2008-08-19 Classification: TRANSFERASE Ligands: SM5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-08-19
Ligands: SM5
