Search Count: 32
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Structure Of Crbn:Ikzf2:Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-09-03 Classification: IMMUNE SYSTEM Ligands: A1CBH, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: A1CBH, ZN
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Structure Of Crbn:Ikzf2:Compound 35
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2025-09-03 Classification: IMMUNE SYSTEM Ligands: A1CBG, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: A1CBG, ZN
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Structure Of Ikzf2:Crbn:Compound 5 Ternary Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2025-07-09 Classification: IMMUNE SYSTEM Ligands: A1CAC, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-09
Ligands: A1CAC, ZN
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Structure Of Crbn Tbd Bound To Compound C1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2025-05-28 Classification: IMMUNE SYSTEM Ligands: A1CAV, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1CAV, ZN
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Structure Of Crbn Tbd Bound To Compound C3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2025-05-28 Classification: IMMUNE SYSTEM Ligands: A1CAW, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1CAW, ZN
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Pvtx-405: A Potent, Highly Selective, And Orally Efficacious Molecular Glue Degrader Of Ikzf2 For Cancer Immunotherapy
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2025-05-14 Classification: TRANSCRIPTION Ligands: A1A8N, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1A8N, ZN
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Discovery Of Potent, Highly Selective And Efficacious Smarca2 Degraders - Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: A1BF5, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1BF5, ZN
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Discovery Of Potent, Highly Selective And Efficacious Smarca2 Degraders - Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: A1A1O, ZN, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1O, ZN, ACT
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Discovery Of Potent, Highly Selective And Efficacious Smarca2 Degraders - Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: A1A1P, ZN, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1P, ZN, ACT
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Recombinant Ym1 Crystal Structure
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2024-01-17 Classification: IMMUNE SYSTEM Ligands: ACT, GOL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2024-01-17
Ligands: ACT, GOL
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Ex Vivo Ym1 Crystal Structure
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2024-01-17 Classification: IMMUNE SYSTEM Ligands: EDO |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2024-01-17
Ligands: EDO
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Recombinant Ym2 Crystal Structure
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.17 Å Release Date: 2024-01-17 Classification: IMMUNE SYSTEM Ligands: EDO |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2024-01-17
Ligands: EDO
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Ex Vivo Ym2 Crystal Structure
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2024-01-17 Classification: IMMUNE SYSTEM Ligands: GOL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2024-01-17
Ligands: GOL
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: SAH, ZN, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: SAH, ZN, EDO, GOL
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3830052
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, X52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, X52
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3685032A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, UXM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, UXM
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, GOL, SAH, LUP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, GOL, SAH, LUP
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, EDO, SAM, L0J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, EDO, SAM, L0J
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, SAM, O41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, SAM, O41
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, GOL, SAM, O6A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, GOL, SAM, O6A
