Search Count: 4,820
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Crystal Structure Of Epoxomicin:20S Proteasome Reveals A Molecular Basis For Selectivity Of Alpha,Beta-Epoxyketone Proteasome Inhibitors
Organism: Saccharomyces cerevisiae, Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2000-11-27 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: MG |
Organism: Saccharomyces cerevisiae, Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2000-11-27
Ligands: MG
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Bile Salt Hydrolase From B. Longum With Covalent Inhibitor Bound
Organism: Bifidobacterium longum
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2023-11-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: WSR |
Organism: Bifidobacterium longum
Method: X-RAY DIFFRACTION
Release Date: 2023-11-01
Ligands: WSR
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Cryo-Em Structure Of Human P97/Vcp Bound To Inhibitor Gnd-135
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2026-05-27 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ADP, A1CBF |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-05-27
Ligands: ADP, A1CBF
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Crystal Structure Of Sars-Cov-2 3Cl Protease In Complex With Inhibitor Psr-I-162
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2026-06-10 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2026-06-10
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Crystal Structure Of Sars-Cov-2 3Cl Protease In Complex With Inhibitor Amj-Ii-122
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2026-06-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: A1C2R, PG4 |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2026-06-10
Ligands: A1C2R, PG4
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Crystal Structure Of Sars-Cov-2 3Cl Protease In Complex With Inhibitor Amj-Ii-72
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2026-06-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: A1C2N, PG4 |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2026-06-10
Ligands: A1C2N, PG4
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Crystal Structure Of Sars-Cov-2 3Cl Protease In Complex With Inhibitor Nn-Iv-169
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2026-06-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: A1C2Q, BR |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2026-06-10
Ligands: A1C2Q, BR
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Crystal Structure Of Sars-Cov-2 3Cl Protease In Complex With Inhibitor Csd-V-169
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2026-06-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: A1C4H, PEG, CL, PG4 |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2026-06-10
Ligands: A1C4H, PEG, CL, PG4
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Room Temperature X-Ray Structure Of Sars Cov-2 Main Protease Intermediate Precursor With Ensitrelvir (Esv)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2026-05-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 7YY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-06
Ligands: 7YY
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z1530301542
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: CIT, ZQA |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-06-09
Ligands: CIT, ZQA
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z1673618163
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: WL7 |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-06-09
Ligands: WL7
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z319891284
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: CIT, ZQD |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-06-09
Ligands: CIT, ZQD
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z68299550
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: JOV |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-06-09
Ligands: JOV
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With En300-100112
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: ZQJ |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-06-09
Ligands: ZQJ
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With En300-321461
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: CIT, WOY |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-06-09
Ligands: CIT, WOY
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z2697514548
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: GWG |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-06-09
Ligands: GWG
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With En300-1605072
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: ZQG |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-06-09
Ligands: ZQG
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z239136710
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: K3A |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-06-09
Ligands: K3A
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z2856434783
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: O3G |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-06-09
Ligands: O3G
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z31504642
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: CIT, WJD |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-06-09
Ligands: CIT, WJD
