Search Count: 21
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Crystal Structure Of Tead1-Ybd In Complex With Irreversible Compound Swtx-143
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2023-10-04 Classification: TRANSCRIPTION Ligands: K46 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-04
Ligands: K46
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Human Glucokinase In Complex With Novel Indazole Activator.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2017-05-31 Classification: transferase/transferase activator Ligands: GLC, 8WM, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: GLC, 8WM, IOD
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Human Glucokinase In Complex With Novel Pyrazole Activator.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2017-05-31 Classification: transferase/transferase activator Ligands: GLC, 8WJ, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: GLC, 8WJ, IOD
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Crystal Structure Of Carbonmonoxy Hemoglobin S (Liganded Sickle Cell Hemoglobin) Complexed With Gbt Compound 31
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-02-22 Classification: OXYGEN TRANSPORT Ligands: HEM, CMO, 7SJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: HEM, CMO, 7SJ
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Crystal Structure Of Carbonmonoxy Hemoglobin S (Liganded Sickle Cell Hemoglobin) Complexed With Gbt Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2017-02-22 Classification: OXYGEN TRANSPORT Ligands: HEM, CMO, 86M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: HEM, CMO, 86M
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Human Glucokinase In Complex With Novel Activator (2S)-3-Cyclohexyl-2-(6-Fluoro-4-Oxoquinazolin-3(4H)-Yl)-N-(1,3-Thiazol-2-Yl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2013-03-20 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: GLC, 1FW, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: GLC, 1FW, IOD
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Human Glucokinase In Complex With Novel Activator (2S)-3-Cyclohexyl-2-(6-Fluoro-2,4-Dioxo-1,4-Dihydroquinazolin-3(2H)-Yl)-N-(1,3-Thiazol-2-Yl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2013-03-20 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: GLC, 1FX, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: GLC, 1FX, IOD
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Human Glucokinase In Complex With Novel Activator (2S)-3-Cyclohexyl-2-[4-(Methylsulfonyl)-2-Oxopiperazin-1-Yl]-N-(1,3-Thiazol-2-Yl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2013-03-20 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: GLC, 1FY, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: GLC, 1FY, IOD
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Crystal Structure Of Human Dipeptidyl Peptidase Iv In Complex With A Pyridopyrimidinedione Analogue
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-02-27 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0WG, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-27
Ligands: 0WG, NAG
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With Tak-322
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2010-02-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, T22 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: NAG, T22
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With A Pyrimidinedione Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2010-02-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: RUF, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: RUF, NAG
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With A Pyrimidinedione Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2010-02-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: XIH, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: XIH, NAG
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With A Pyrimidinone Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2010-02-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: RUM, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: RUM, NAG
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Crystal Structure Of Human Dpp4 In Complex With A Benzimidazole Derivative
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2008-10-21 Classification: HYDROLASE Ligands: NAG, B2Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-21
Ligands: NAG, B2Y
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Crystal Structure Of Human Dpp4 In Complex With A Benzimidazole Derivative
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2008-10-21 Classification: HYDROLASE Ligands: NAG, 7AC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-21
Ligands: NAG, 7AC
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Crystal Structure Of Human Dpp-4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2008-03-04 Classification: HYDROLASE Ligands: NAG, SY1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-04
Ligands: NAG, SY1
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Structure Of H-Chk1 Complexed With A767085
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: 76A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: 76A
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Structure Of H-Chk1 Complexed With Aa582939
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: A58 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: A58
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Structure Of H-Chk1 Complexed With A771129
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: 77A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: 77A
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Structure Of H-Chk1 Complexed With A780125
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: A25 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: A25
