Search Count: 27
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Crystal Structure Of The P62 Uba Domain Bound To Vhh 6C10
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2025-10-29 Classification: PROTEIN TRANSPORT |
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION
Release Date: 2025-10-29
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Cryo-Em Structure Of Skp1-Fbxo22 In Complex With A Bach1 Btb Dimer At 3.2A Resolution
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Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-12-11
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Cryo-Em Structure Of Skp1-Fbxo22
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Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-12-11
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Homodimer Of Bach1 F9A Mutant Btb Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-12-11 Classification: DNA BINDING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-11
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Homodimer Of Bach1 Btb Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2024-12-11 Classification: DNA BINDING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-11
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Homodimer Of Bach1 Btb Domain In Complex With 2-Methyl-2,4-Pentanediol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2024-12-11 Classification: DNA BINDING PROTEIN Ligands: MRD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-11
Ligands: MRD
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Pi3K Delta In Complex With Sd5
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-05-18 Classification: HYDROLASE Ligands: SD5 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: SD5
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Pi3Kdelta In Complex With An Inhibitor
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2022-05-18 Classification: HYDROLASE Ligands: H5I |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: H5I
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Pi3K Alpha In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2022-05-18 Classification: transferase/inhibitor Ligands: KVJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: KVJ
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Btk In Complex With Lou064, A Potent And Highly Selective Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-03-04 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-04
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Btk In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2019-09-18 Classification: TRANSFERASE Ligands: L0Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-18
Ligands: L0Z
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Discovery Of Cdz173 (Leniolisib), Representing A Structurally Novel Class Of Pi3K Delta-Selective Inhibitors
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2017-09-20 Classification: TRANSFERASE Ligands: 9NQ |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-09-20
Ligands: 9NQ
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Crystal Structure Of Pi3K Alpha With Pi3K Delta Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.02 Å Release Date: 2016-09-07 Classification: Transferase/Protein Transport/Inhibitor Ligands: 6CY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: 6CY
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Discovery Of Imidazoquinolines As A Novel Class Of Potent, Selective And In Vivo Efficacious Cot Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-08-24 Classification: TRANSFERASE Ligands: 6DA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-24
Ligands: 6DA
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Discovery And Pharmacological Characterization Of Novel Quinazoline-Based Pi3K Delta-Selective Inhibitors
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2016-08-10 Classification: TRANSFERASE Ligands: 6CY |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: 6CY
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Serine/Threonine-Protein Kinase Pak1 Complexed With A Dibenzodiazepine: Identification Of An Allosteric Site On Pak1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-08-05 Classification: Transferase/transferase inhibitor Ligands: 4PV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4PV, GOL
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Pak1 In Complex With 2-Chloro-5-Ethyl-8-Fluoro-11-(4-Methylpiperazin-1-Yl)-Dibenzodiazepine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2015-06-24 Classification: TRANSFERASE Ligands: 4OQ, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: 4OQ, MG
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Pak1 In Complex With (S)-N-(Tert-Butyl)-3-((2-Chloro-5-Ethyl-8-Fluoro-Dibenzodiazepin-11-Yl)Amino)Pyrrolidine-1-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-06-24 Classification: TRANSFERASE Ligands: 4OR, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: 4OR, MG
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Crystal Structure Of Cot Kinase Domain In Complex With 5-(2-Amino-5-(Quinolin-3-Yl)Pyridin-3-Yl)-1,3,4-Oxadiazole-2(3H)-Thione
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2015-05-06 Classification: TRANSFERASE Ligands: 49B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: 49B
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Crystal Structure Of Cot Kinase Domain In Complex With 5-(5-(1H-Indol-3-Yl)-1H-Pyrrolo[2,3-B]Pyridin-3-Yl)-1,3,4-Oxadiazol-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2015-05-06 Classification: TRANSFERASE Ligands: 499 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: 499
