Search Count: 20
![]() |
P70 S6K1 In Complex With Msc2317067A-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2022-07-06 Classification: TRANSFERASE/INHIBITOR Ligands: 1RJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: 1RJ
![]() |
P70 S6K1 In Complex With Msc2363318A-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2022-07-06 Classification: TRANSFERASE/INHIBITOR Ligands: 1SK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: 1SK
![]() |
Btk In Complex With 18A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2021-10-06 Classification: TRANSFERASE/INHIBITOR Ligands: 2IE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 2IE
![]() |
Btk In Complex With 25A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2021-10-06 Classification: TRANSFERASE/INHIBITOR Ligands: 2IJ, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 2IJ, DMS
![]() |
Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9J, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9J, DMS
![]() |
Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9M
![]() |
Btk1 Soaked With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9P, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9P, DMS
![]() |
Btk1 Soaked With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9S, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9S, DMS
![]() |
Btk1 Soaked With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9V, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9V, DMS
![]() |
Btk1 Soaked With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: DMS, X9Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: DMS, X9Y
![]() |
Structure Of Human Bruton'S Tyrosine Kinase In Complex With Evobrutinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2019-08-14 Classification: Transferase/Transferase Inhibitor Ligands: CL, MZJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-14
Ligands: CL, MZJ
![]() |
Discovery Of Affinity-Based Probes For Btk Occupancy Assay
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2019-02-06 Classification: IMMUNE SYSTEM Ligands: KHD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: KHD
![]() |
Crystal Structure Of Btk In Complex With Fragment Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2018-10-17 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: GJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: GJG
![]() |
Crystal Structure Of Btk In Complex With Covalent Fragment Ligand
Organism: homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2018-10-17 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: GJD |
Organism: homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: GJD
![]() |
Crystal Structure Of Btk In Complex With Fragment Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-09-05 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: GJA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: GJA
![]() |
Crystal Structure Of Btk In Complex With Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2018-09-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GJ7, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: GJ7, DMS
![]() |
Crystal Structure Of Btk In Complex With Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2018-09-05 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: GJJ, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: GJJ, DMS
![]() |
Structure Of Follicle-Stimulating Hormone In Complex With The Entire Ectodomain Of Its Receptor (P31)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2014-04-09 Classification: SIGNALING PROTEIN Ligands: NAG, EDO, JEF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-09
Ligands: NAG, EDO, JEF
![]() |
Crystal Structure Of Aurora Kinase A In Complex With N-{4-[(6-Oxo-5,6-Dihydrobenzo[C][1,8]Naphthyridin-1-Yl)Amino]Phenyl}Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2013-05-22 Classification: transferase/transferase inhibitor Ligands: XU2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: XU2
![]() |
Crystal Structure Of Aurora Kinase A In Complex With Benzo[C][1,8]Naphthyridin-6(5H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2013-05-22 Classification: transferase/transferase inhibitor Ligands: XU1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: XU1
