Search Count: 19
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Crystal Structure Of Crystal Form 2 Of An Active Kras G12D (Gppcp) Dimer In Complex With Bi-5747
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2020-11-18 Classification: SIGNALING PROTEIN Ligands: MG, GCP, R6W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: MG, GCP, R6W
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Crystal Structure Of Gmppnp-Bound G12R Mutant Of Human Kras4B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-09-25 Classification: ONCOPROTEIN Ligands: MG, GNP, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: MG, GNP, GOL
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Crystal Structure Of Kras G12D (Gppcp) In Complex With 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: GCP, MG, F0N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: GCP, MG, F0N
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Crystal Structure Of Kras G12D (Gppcp) In Complex With 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: MG, NO3, GCP, EZZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: MG, NO3, GCP, EZZ
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Crystal Structure Of Kras G12D (Gppcp) In Complex With 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: MG, GCP, F0B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: MG, GCP, F0B
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Crystal Structure Of Kras G12D (Gppcp) In Complex With Bi 2852
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: F0K, MG, GCP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: F0K, MG, GCP
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Discovery Of Potent Myeloid Cell Leukemia-1 (Mcl-1) Inhibitors Using Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-01-18 Classification: apoptosis/apoptosis inhibitor Ligands: 6AL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-18
Ligands: 6AL
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Discovery Of Potent Myeloid Cell Leukemia-1 (Mcl-1) Inhibitors Using Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2017-01-18 Classification: apoptosis/apoptosis inhibitor Ligands: 6AK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-18
Ligands: 6AK
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Mcl-1 Complexed With Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2016-03-02 Classification: apoptosis/apoptosis inhibitor Ligands: 5WL, 5WK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-02
Ligands: 5WL, 5WK
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Mcl-1 Complexed With Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-03-02 Classification: apoptosis/apoptosis inhibitor Ligands: 5X2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-02
Ligands: 5X2
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Mcl-1 Complexed With Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-03-02 Classification: APOPTOSIS/APOPTOSIS inhibitor Ligands: 5X3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-02
Ligands: 5X3
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X-Ray Crystal Structure Of Ns3 Helicase From Hcv With A Bound Fragment Inhibitor At 2.08 A Resolution
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2015-12-23 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2015-12-23
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X-Ray Crystal Structure Of Ns3 Helicase From Hcv With A Bound Inhibitor At 2.42 A Resolution
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2015-12-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 3VZ |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2015-12-23
Ligands: 3VZ
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Mcl-1 Complexed With Small Molecules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-04-29 Classification: apoptosis/apoptosis inhibitor Ligands: 4M7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-29
Ligands: 4M7
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Mcl-1 Complexed With Small Molecules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-04-29 Classification: apoptosis/apoptosis inhibitor Ligands: 4M6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-29
Ligands: 4M6
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X-Ray Crystal Structure Of Human Alpha-Thrombin With A Tripeptide Phosphonate Inhibitor.
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2001-03-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: PHV |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 2001-03-02
Ligands: PHV
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X-Ray Structure Of The Human Alpha-Thrombin Complex With A Tripeptide Phosphonate Inhibitor.
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2001-02-26 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: PHW |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 2001-02-26
Ligands: PHW
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Complex Of Human Alpha-Thrombin With The Bifunctional Boronate Inhibitor Borolog1
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 1998-06-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: T29 |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 1998-06-03
Ligands: T29
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Complex Of Human Alpha-Thrombin With The Bifunctional Boronate Inhibitor Borolog2
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 1998-06-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: T16 |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 1998-06-03
Ligands: T16
