Search Count: 30
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Hiv-Rt Pre-Catalytic Complex With Mk-8527
Organism: Hiv-1 m:b_hxb2r, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2025-09-17 Classification: TRANSFERASE/DNA Ligands: MG, A1A6R |
Organism: Hiv-1 m:b_hxb2r, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2025-09-17
Ligands: MG, A1A6R
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Crystal Structure Of Catalytic Domain Of Tace With 2-(2-Aminothiazol-4-Yl)Pyrrolidine-Based Tartrate Diamides
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2011-04-20 Classification: hydrolase/hydrolase inhibitor Ligands: IPA, INN, ZN, CA, 786 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-20
Ligands: IPA, INN, ZN, CA, 786
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Hcv Ns3-4A Protease Domain With A Ketoamide Inhibitor Derivative Of Boceprevir Bound
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2011-02-23 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, MCX, BME |
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION
Release Date: 2011-02-23
Ligands: ZN, MCX, BME
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Hcv Ns3-4A Protease Domain With Ketoamide Inhibitor Narlaprevir
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-01-19 Classification: VIRAL PROTEIN/INHIBITOR Ligands: ZN, NNA, BME |
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION
Release Date: 2011-01-19
Ligands: ZN, NNA, BME
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Hcv Ns3 Protease Domain With P1-P3 Macrocyclic Ketoamide Inhibitor
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2010-10-27 Classification: VIRAL PROTEIN Ligands: ZN, JZT, BME |
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: ZN, JZT, BME
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Crystal Structure Of Catalytic Domain Of Tace With Benzimidazolyl-Thienyl-Tartrate Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-07-28 Classification: HYDROLASE Ligands: ZN, 50X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-28
Ligands: ZN, 50X
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Crystal Structure Of Catalytic Domain Of Tace With Hydantoin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2010-03-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, INN, IPA, Z94 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: ZN, INN, IPA, Z94
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Crystal Structure Of Catalytic Domain Of Tace With The First Hydantoin Inhibitor Occupying The S1' Pocket
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2010-03-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, 724 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: ZN, 724
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Discovery Of C-Imidazole Azaheptapyridine Fpt Inhibitors
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-01-26 Classification: TRANSFERASE Ligands: MG, ZN, FPP, Z96 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2010-01-26
Ligands: MG, ZN, FPP, Z96
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Hcv Ns3 Protease Domain With Ketoamide Inhibitor
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2010-01-19 Classification: HYDROLASE Ligands: ZN, M66 |
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION
Release Date: 2010-01-19
Ligands: ZN, M66
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Crystal Structure Of Catalytic Domain Of Tace With Tartrate-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2009-12-22 Classification: HYDROLASE Ligands: ZN, INN, 403 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-22
Ligands: ZN, INN, 403
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Crystal Structure Of Catalytic Domain Of Tace With Phenyl-Pyrrolidinyl-Tartrate Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2009-12-22 Classification: HYDROLASE Ligands: ZN, INN, IPA, Z59 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-22
Ligands: ZN, INN, IPA, Z59
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Structure Of Hcv Ns3-4A Protease With An Inhibitor Derived From A Boronic Acid
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2009-02-10 Classification: VIRAL PROTEIN Ligands: ZN, BE8 |
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION
Release Date: 2009-02-10
Ligands: ZN, BE8
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Crystal Structure Of The S139A Mutant Of Hepatitis C Virus Ns3/4A Protease
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2007-10-09 Classification: VIRAL PROTEIN Ligands: ZN, NA |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2007-10-09
Ligands: ZN, NA
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Structure Of Hepatitis C Viral Ns3 Protease Domain Complexed With Ns4A Peptide And Ketoamide Sch476776
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2007-07-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, BME, HUD |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2007-07-31
Ligands: ZN, BME, HUD
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Discovery Of The Hcv Ns3/4A Protease Inhibitor Sch503034. Key Steps In Structure-Based Optimization
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-07-31 Classification: VIRAL PROTEIN Ligands: ZN |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2007-07-31
Ligands: ZN
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Structure Of Ns3 Complexed With A Ketoamide Inhibitor Sch491762
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2007-07-31 Classification: VIRAL PROTEIN Ligands: ZN, BME, HU1 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2007-07-31
Ligands: ZN, BME, HU1
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Structure Of The Hcv Ns3/4A Protease Inhibitor Cvs4819
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2007-07-31 Classification: VIRAL PROTEIN Ligands: ZN, HU2 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2007-07-31
Ligands: ZN, HU2
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Structure Of Hepatitis C Viral Ns3 Protease Domain Complexed With Ns4A Peptide And Ketoamide Sch571696
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2007-07-31 Classification: VIRAL PROTEIN Ligands: ZN, BME, HU4 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2007-07-31
Ligands: ZN, BME, HU4
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Structure Of Hepatitis C Viral Ns3 Protease Domain Complexed With Ns4A Peptide And Ketoamide Sch503034
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2007-07-31 Classification: VIRAL PROTEIN Ligands: ZN, BME, U5G |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2007-07-31
Ligands: ZN, BME, U5G
