Search Count: 16
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Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 1.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: GQD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: GQD
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Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 2.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: QHG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: QHG
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Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 3.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: J0W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: J0W
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Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 4.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: 7QN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: 7QN
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Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 5.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: VQI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: VQI
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A Novel Oral Selective Estrogen Receptor Down-Regulator, Azd9496, Drives Tumour Growth Inhibition In Estrogen Receptor Positive And Esr1 Mutant Models
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2015-12-16 Classification: SIGNALING PROTEIN Ligands: KE9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: KE9
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Discovery Of Pyrimidine Isoxazoles Inha In Complex With Compound 6
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2015-09-30 Classification: OXIDOREDUCTASE Ligands: NAD, MG, HRW |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: NAD, MG, HRW
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Discovery Of Pyrimidine Isoxazoles Inha In Complex With Compound 9
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2015-09-30 Classification: OXIDOREDUCTASE Ligands: NAD, MG, KI5 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: NAD, MG, KI5
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Discovery Of Pyrimidine Isoxazoles Inha In Complex With Compound 15
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2015-09-30 Classification: OXIDOREDUCTASE Ligands: NAD, MG, 1PE, A0C |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: NAD, MG, 1PE, A0C
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Discovery Of Pyrimidine Isoxazoles Inha In Complex With Compound 10
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2015-09-30 Classification: OXIDOREDUCTASE Ligands: NAD, UUD, ACT |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: NAD, UUD, ACT
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Discovery Of Pyrimidine Isoxazoles Inha In Complex With Compound 23
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2015-09-30 Classification: OXIDOREDUCTASE Ligands: NAD, KXU |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: NAD, KXU
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Crystal Structure Of Inha(S94A) Mutant In Complex With Pyridomycin
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2013-12-04 Classification: OXIDOREDUCTASE Ligands: PYW |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2013-12-04
Ligands: PYW
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Crystal Structure Of Inha(S94A) Mutant In Complex With Oh-141
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2013-12-04 Classification: OXIDOREDUCTASE Ligands: I4I, NAD |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2013-12-04
Ligands: I4I, NAD
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How Nature Bridges The Gap: Crystallographic Elucidation Of Pyridomycin Binding To Inha
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2013-12-04 Classification: OXIDOREDUCTASE Ligands: NAD, PYW |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2013-12-04
Ligands: NAD, PYW
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Alk5 In Complex With 4-((5,6-Dimethyl-2-(2-Pyridyl)-3-Pyridyl)Oxy)-N-(3,4,5-Trimethoxyphenyl)Pyridin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2009-09-22 Classification: TRANSFERASE Ligands: ZZG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-09-22
Ligands: ZZG, EDO
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Alk5 In Complex With 4-((4-((2,6-Dimethyl-3-Pyridyl)Oxy)-2-Pyridyl) Amino)Benzenesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2009-09-22 Classification: TRANSFERASE Ligands: EDO, ZZF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-09-22
Ligands: EDO, ZZF
