Search Count: 13
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Crystal Structure Of Tyrosine Kinase 2 Jh2 (Pseudo Kinase Domain) Complexed With Compound-12 Aka:6-[(Cyclopropanecarbonyl)Amino]-4-{[2-Methoxy-3-(Pyrimidin-2-Yl)Phenyl]Amino}-N-Methylpyridazine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2021-08-04 Classification: TRANSFERASE Ligands: VZJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-04
Ligands: VZJ
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Crystal Structure Of Tyrosine Kinase 2 Jh2 (Pseudo Kinase Domain) Complexed With Compound-12 Aka:6-[(Cyclopropanecarbonyl)Amino]-4-({3-[6-(Dimethylcarbamoyl)Pyridazin-3-Yl]-2-Methoxyphenyl}Amino)-N-Methylpyridazine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2021-08-04 Classification: TRANSFERASE Ligands: VZG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-04
Ligands: VZG
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Btk In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2019-04-03 Classification: TRANSFERASE/INHIBITOR Ligands: LTJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-03
Ligands: LTJ
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Crystal Structure Of Pi3K Delta In Complex With A Trifluoro-Ethyl-Pyrazol-Pyrolotriazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-06-07 Classification: TRANSFERASE/TRANSFERASE REGULATOR Ligands: 9EM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: 9EM
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Crystal Structure Of Bruton Agammabulinemia Tyrosine Kinase Complexed With Bms-986142 Aka (2S)-6-Fluoro-5-[3-(8-Fluoro-1-Methyl-2,4-Dioxo-1,2,3,4-Tetrahydroquinazolin-3-Yl)-2-Methylphenyl]-2-(2-Hydroxypropan-2-Yl)-2,3,4,9-Tetrahydro-1H-Carbazole-8-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2017-03-08 Classification: TRANSFERASE Ligands: 73T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-08
Ligands: 73T
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P38 Alpha Kinase Complexed With A Pyrazolo-Triazine Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2012-02-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: NK0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-01
Ligands: NK0
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P38 Alpha Map Kinase Complexed With Pyrrolotriazine Inhibitor 7K
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2010-10-13 Classification: TRANSFERASE Ligands: 38P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: 38P
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P38 Alpha Map Kinase Complexed With Pyrrolotriazine Inhibitor 7V
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-10-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 39P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: 39P
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Morpholino Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2008-04-15 Classification: TRANSFERASE Ligands: P39 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-15
Ligands: P39
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P38 Alpha Map Kinase Complexed With Bms-640994
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-04-15 Classification: SIGNALING PROTEIN, TRANSFERASE Ligands: 304 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-15
Ligands: 304
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Morpholino Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-04-08 Classification: TRANSFERASE Ligands: P38 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-08
Ligands: P38
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Phenylalanine Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 11B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: 279 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: 279
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Phenylalanine Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 11J
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: 287 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: 287
