Search Count: 33
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B-Raf Kinase V600E Oncogenic Mutant In Complex With Plx3203
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2012-08-08 Classification: Transferase/Transferase inhibitor Ligands: 325 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: 325
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B-Raf Kinase In Complex With Plx4720
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2008-02-26 Classification: TRANSFERASE Ligands: 324 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-02-26
Ligands: 324
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Pim-1 Kinase Domain In Complex With 3-Aminophenyl-7-Azaindole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2008-02-26 Classification: TRANSFERASE Ligands: IMD, C4E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-02-26
Ligands: IMD, C4E
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Fgfr Tyrosine Kinase Domain In Complex With 3-(3-Methoxybenzyl)-7-Azaindole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2008-02-26 Classification: TRANSFERASE Ligands: C4F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-02-26
Ligands: C4F
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Catalytic Domain Of Human Phosphodiesterase 4D In Complex With 3,5-Dimethyl-1H-Pyrazole-4-Carboxylic Acid Ethyl Ester
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2005-03-01 Classification: HYDROLASE Ligands: ZN, MG, DEE, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
Ligands: ZN, MG, DEE, EDO
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Catalytic Domain Of Human Phosphodiesterase 4D In Complex With 3,5-Dimethyl-1-Phenyl-1H-Pyrazole-4-Carboxylic Acid Ethyl Ester
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2005-03-01 Classification: HYDROLASE Ligands: ZN, MG, 3DE, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
Ligands: ZN, MG, 3DE, EDO
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Catalytic Domain Of Human Phosphodiesterase 4D In Complex With 1-(4-Methoxy-Phenyl)-3,5-Dimethyl-1H-Pyrazole-4-Carboxylic Acid Ethyl Ester
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2005-03-01 Classification: HYDROLASE Ligands: ZN, MG, 4DE, EDO, B3P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
Ligands: ZN, MG, 4DE, EDO, B3P
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Catalytic Domain Of Human Phosphodiesterase 4D In Complex With 1-(4-Amino-Phenyl)-3,5-Dimethyl-1H-Pyrazole-4-Carboxylic Acid Ethyl Ester
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2005-03-01 Classification: HYDROLASE Ligands: ZN, MG, 5DE, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
Ligands: ZN, MG, 5DE, EDO
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Catalytic Domain Of Human Phosphodiesterase 4B In Complex With 1-(2-Chloro-Phenyl)-3,5-Dimethyl-1H-Pyrazole-4-Carboxylic Acid Ethyl Ester
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2005-03-01 Classification: HYDROLASE Ligands: ZN, MG, 6DE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
Ligands: ZN, MG, 6DE
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Catalytic Domain Of Human Phosphodiesterase 4B In Complex With 3,5-Dimethyl-1-(3-Nitro-Phenyl)-1H-Pyrazole-4-Carboxylic Acid Ethyl Ester
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2005-03-01 Classification: HYDROLASE Ligands: ZN, MG, 7DE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
Ligands: ZN, MG, 7DE
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Catalytic Domain Of Human Phosphodiesterase 4D In Complex With 3,5-Dimethyl-1-(3-Nitro-Phenyl)-1H-Pyrazole-4-Carboxylic Acid Ethyl Ester
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.36 Å Release Date: 2005-03-01 Classification: HYDROLASE Ligands: ZN, MG, 7DE, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
Ligands: ZN, MG, 7DE, EDO
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Catalytic Domain Of Human Phosphodiesterase 4B In Complex With Cilomilast
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2004-12-14 Classification: HYDROLASE Ligands: ZN, MG, CIO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-12-14
Ligands: ZN, MG, CIO
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Catalytic Domain Of Human Phosphodiesterase 4B In Complex With Filaminast
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2004-12-14 Classification: HYDROLASE Ligands: ZN, MG, FIL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-12-14
Ligands: ZN, MG, FIL
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Catalytic Domain Of Human Phosphodiesterase 4B In Complex With Piclamilast
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2004-12-14 Classification: HYDROLASE Ligands: ZN, MG, PIL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-12-14
Ligands: ZN, MG, PIL
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Catalytic Domain Of Human Phosphodiesterase 4B In Complex With (R)-Mesopram
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2004-12-14 Classification: HYDROLASE Ligands: ZN, MG, 5RM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-12-14
Ligands: ZN, MG, 5RM
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Catalytic Domain Of Human Phosphodiesterase 4B In Complex With Roflumilast
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2004-12-14 Classification: HYDROLASE Ligands: ZN, MG, ROF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-12-14
Ligands: ZN, MG, ROF
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Catalytic Domain Of Human Phosphodiesterase 4B In Complex With (R)-Rolipram
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2004-12-14 Classification: HYDROLASE Ligands: ZN, MG, ROL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-12-14
Ligands: ZN, MG, ROL
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Catalytic Domain Of Human Phosphodiesterase 4B In Complex With (R,S)-Rolipram
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2004-12-14 Classification: HYDROLASE Ligands: ZN, MG, ROL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-12-14
Ligands: ZN, MG, ROL
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Catalytic Domain Of Human Phosphodiesterase 4D In Complex With Cilomilast
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2004-12-14 Classification: HYDROLASE Ligands: ZN, MG, CIO, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-12-14
Ligands: ZN, MG, CIO, EDO
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Catalytic Domain Of Human Phosphodiesterase 4D In Complex With Piclamilast
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2004-12-14 Classification: HYDROLASE Ligands: ZN, MG, PIL, B3P, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-12-14
Ligands: ZN, MG, PIL, B3P, EDO
