Search Count: 7
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Structure-Based Discovery Of Novel Non-Covalent Small Molecule Inhibitors Of Usp30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2025-05-21 Classification: HYDROLASE Ligands: A1L7W, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-21
Ligands: A1L7W, ZN
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Identification Of Small-Molecule Binding Sites Of A Ubiquitin-Conjugating Enzyme-Ube2T Through Fragment-Based Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2024-02-28 Classification: LIGASE Ligands: V23, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-28
Ligands: V23, EDO
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Identification Of Small-Molecule Binding Sites Of A Ubiquitin-Conjugating Enzyme-Ube2T Through Fragment-Based Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2024-02-28 Classification: LIGASE Ligands: V2R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-28
Ligands: V2R
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Identification And Characterization Of Inhibitors Covalently Modifying Catalytic Cysteine Of Ube2T And Blocking Ubiquitin Transfer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2023-11-29 Classification: LIGASE/INHIBITOR Ligands: V6C, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-29
Ligands: V6C, EDO
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Identification And Characterization Of Inhibitors Covalently Modifying Catalytic Cysteine Of Ube2T And Blocking Ubiquitin Transfer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2023-11-29 Classification: LIGASE/INHIBITOR Ligands: V5L, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-29
Ligands: V5L, EDO
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Crystal Structure Of Smyd3 In Complex With Covalent Inhibitor 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2019-08-14 Classification: TRANSFERASE/INHIBITOR Ligands: A8U, ZN, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-14
Ligands: A8U, ZN, SAM
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Crystal Structure Of Smyd3 In Complex With Covalent Inhibitor 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2018-10-17 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, 8W0, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: ZN, 8W0, SAM
