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Search Count: 22

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6P8W image
Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.

6P8X image
Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.

6P8Y image
Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.

6P8Z image
Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor

2ZJH image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-(1-Benzyl-Piperidin-4-Yl)-4-Mercapto-Butyramide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.60 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1H

2ZJI image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-[1-(2,6-Dimethoxy-Benzyl)-Piperidin-4-Yl]-4-Mercapto-Butyramide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1I

2ZJJ image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With 4-(4-Fluoro-Benzyl)-Piperazine-2-Carboxylic Acid (2-Mercapto-Ethyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1J

2ZJK image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With 4-(4-Fluoro-Benzyl)-Piperazine-2-Carboxylic Acid(3-Mercapto-Propyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.00 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1K

2ZJL image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-[1-(5-Bromo-2,3-Dimethoxy-Benzyl)-Piperidin-4-Yl]-4-Mercapto-Butyramide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1L

2ZJM image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-[1-(5-Chloro-2-Isopropoxy-3-Methoxy-Benzyl)-Piperidin-4-Yl]-2-(4-Sulfamoyl-Phenoxy)-Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1M

2ZJN image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-[1-(5-Chloro-2-Isopropoxy-3-Methoxy-Benzyl)-Piperidin-4-Yl]-2-(2-Methyl-4-Sulfamoyl-Phenoxy)-Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1N

3DB8 image
Crystal Structure Of An Activated (Thr->Asp) Polo-Like Kinase 1 (Plk1) Catalytic Domain In Complex With Compound 041
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Resolution:3.15 Å Release Date: 2008-10-07
Classification: TRANSFERASE
Ligands: 1FR

3DBC image
Crystal Structure Of An Activated (Thr->Asp) Polo-Like Kinase 1 (Plk1) Catalytic Domain In Complex With Compound 257
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Resolution:3.35 Å Release Date: 2008-10-07
Classification: TRANSFERASE
Ligands: 2FR

3DBD image
Crystal Structure Of An Activated (Thr->Asp) Polo-Like Kinase 1 (Plk1) Catalytic Domain In Complex With Compound 094
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Resolution:3.05 Å Release Date: 2008-10-07
Classification: TRANSFERASE
Ligands: 3FR

3DBE image
Crystal Structure Of An Activated (Thr->Asp) Polo-Like Kinase 1 (Plk1) Catalytic Domain In Complex With Compound 557
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Resolution:3.32 Å Release Date: 2008-10-07
Classification: TRANSFERASE
Ligands: 4FR

3DBF image
Crystal Structure Of An Activated (Thr->Asp) Polo-Like Kinase 1 (Plk1) Catalytic Domain In Complex With Compound 562
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Resolution:3.20 Å Release Date: 2008-10-07
Classification: TRANSFERASE
Ligands: 5FR

3D5U image
Crystal Structure Of A Wildtype Polo-Like Kinase 1 (Plk1) Catalytic Domain.

3D5V image
Crystal Structure Of An Activated (Thr->Asp) Polo-Like Kinase 1 (Plk1) Catalytic Domain.

3D5W image
Crystal Structure Of A Phosphorylated Polo-Like Kinase 1 (Plk1) Catalytic Domain In Complex With Adp.
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Resolution:2.60 Å Release Date: 2008-08-26
Classification: TRANSFERASE
Ligands: ADP

3D5X image
Crystal Structure Of An Activated (Thr->Asp) Polo-Like Kinase 1 (Plk1) Catalytic Domain In Complex With Wortmannin.
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2008-08-26
Classification: TRANSFERASE
Ligands: KWT
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