Structural Entry Filters:

Search Count: 24

All Selected
9R0D image
Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2025-11-12
Classification: HYDROLASE
Ligands: ZN, CA, NAG, A1JCF, PO4

9R0G image
Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.43 Å Release Date: 2025-11-12
Classification: HYDROLASE
Ligands: ZN, CA, NAG, A1JCG, PO4

9R0H image
Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 6 (Oric-533)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.28 Å Release Date: 2025-11-12
Classification: HYDROLASE
Ligands: ZN, CA, A1JCH, PO4

9U8C image
Crystal Structure Of Egfr Exon20 Insertion Mutant In Complex With Enozertinib (Oric-114)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.50 Å Release Date: 2025-11-12
Classification: SIGNALING PROTEIN
Ligands: A1L8T

8EXL image
Crystal Structure Of Pi3K-Alpha In Complex With Taselisib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.99 Å Release Date: 2022-11-30
Classification: CELL CYCLE
Ligands: 799

8EXO image
Crystal Structure Of Pi3K-Alpha In Complex With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.46 Å Release Date: 2022-11-30
Classification: CELL CYCLE
Ligands: X3W

8EXU image
Crystal Structure Of Pi3K-Alpha In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.68 Å Release Date: 2022-11-30
Classification: CELL CYCLE
Ligands: X3R

8EXV image
Crystal Structure Of Pi3K-Alpha In Complex With Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.48 Å Release Date: 2022-11-30
Classification: CELL CYCLE
Ligands: X3N

7MSA image
Gdc-9545 In Complex With Estrogen Receptor Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.24 Å Release Date: 2021-06-02
Classification: TRANSCRIPTION
Ligands: G9J, ZNM

7JV8 image
Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 35
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.46 Å Release Date: 2020-09-23
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: ZN, CA, VPD

7JV9 image
Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2020-09-23
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: ZN, CA, NAG, VPG, PO4

6WOK image
Crystal Structure Of Estrogen Receptor Alpha In Complex With Receptor Degrader 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.31 Å Release Date: 2020-07-01
Classification: NUCLEAR PROTEIN
Ligands: G9J, U6D

4O0R image
Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2014-02-12
Classification: transferase/transferase inhibitor
Ligands: 7KC

4O0T image
Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.60 Å Release Date: 2014-02-12
Classification: transferase/transferase inhibitor
Ligands: 2OL

4O0V image
Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2014-02-12
Classification: transferase/transferase inhibitor
Ligands: 2OL

4O0X image
Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.48 Å Release Date: 2014-02-12
Classification: transferase/transferase inhibitor
Ligands: 2OQ

4O0Y image
Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2014-02-12
Classification: transferase/transferase inhibitor
Ligands: 2OO

4LMN image
Crystal Structure Of Mek1 Kinase Bound To Gdc0973
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2013-08-07
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: ANP, MG, EUI

4EKK image
Akt1 With Amp-Pnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2012-05-23
Classification: TRANSFERASE
Ligands: ANP, MN

4EKL image
Akt1 With Gdc0068
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2012-05-23
Classification: TRANSFERASE
Ligands: 0RF
Protein Functional Filters:
Feedback Form
Name
Email
Institute
Feedback