Search Count: 15
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Crystal Structure Of Bcl-Xl In Complex With A Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2024-10-16 Classification: APOPTOSIS Ligands: A1AFG, CD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-16
Ligands: A1AFG, CD
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Crystal Structure Of The Mertk Kinase Domain With Sa4488
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2024-10-09 Classification: TRANSFERASE Ligands: A1APF, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1APF, CL
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Mertk In Complex With Small Molecule 6-{1-[([1,1'-Biphenyl]-4-Yl)Carbamoyl]Azetidin-3-Yl}-3-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]Pyrazine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2024-10-09 Classification: TRANSFERASE/INHIBITOR Ligands: A1APG, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1APG, CL
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Mertk In Complex With Small Molecule Inhibitor 6-{1-[6-(3-Hydroxy-3-Methylbutoxy)-1,3-Benzoxazol-2-Yl]Azetidin-3-Yl}-3-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]Pyrazine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2024-10-09 Classification: TRANSFERASE/INHIBITOR Ligands: A1APH, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1APH, CL
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Crystal Structure Of Bcl-Xl In Complex With Tetrahydroisoquinoline-Pyridine Based Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-10-21 Classification: APOPTOSIS/APOPTOSIS INHIBITOR Ligands: RQ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-21
Ligands: RQ7
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The Novel P300/Cbp Inhibitor A-485 Uncovers A Unique Mechanism Of Action To Target Ar In Castrate Resistant Prostate Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-09-27 Classification: transferase/transferase INHIBITOR Ligands: 6TF, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: 6TF, NA
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Brd4_Bd2-A-35165
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2017-06-28 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 89J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 89J
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Crystal Structure Of Human Nampt With Isoindoline Urea Inhibitor Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8HY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 8HY
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Crystal Structure Of Human Nampt With Isoindoline Urea Inhibitor Compound 53
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8HV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 8HV
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Brd4_Bd2_A-1107604
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 0S6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 0S6
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Brd2 Bromodomain2 With A-1360579
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 87D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 87D
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Brd4_Bd2_A-1497627
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 89D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 89D
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Brd4_Bd2_A-1412838
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 88M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 88M
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Brd4_Bd2_A-1342843
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 89G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 89G
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Solution Structure Of Csra, A Bacterial Carbon Storage Regulatory Protein
Organism: Bacillus subtilis
Method: SOLUTION NMR Release Date: 2005-10-18 Classification: RNA BINDING PROTEIN |
Organism: Bacillus subtilis
Method: SOLUTION NMR
Release Date: 2005-10-18
