Structural Entry Filters:

Search Count: 16

All Selected
6XRN image
Crystal Structure Of Human Pi3K-Gamma In Complex With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.96 Å Release Date: 2021-11-03
Classification: TRANSFERASE/TRANSFERASE inhibitor
Ligands: V84

6XRL image
Crystal Structure Of Human Pi3K-Gamma In Complex With Inhibitor Ipi-549
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.99 Å Release Date: 2020-09-16
Classification: TRANSFERASE/TRANSFERASE inhibitor
Ligands: V7Y, SO4

6XRM image
Crystal Structure Of Human Pi3K-Gamma In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.88 Å Release Date: 2020-09-16
Classification: TRANSFERASE/TRANSFERASE inhibitor
Ligands: V81, SO4

6Z9D image
Human Ecto-5'-Nucleotidase (Cd73) In Complex With Aopcp Derivative Ab680 (Compound 55 In Publication) In The Closed Form (Crystal Form Iii)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2020-09-16
Classification: HYDROLASE
Ligands: ZN, CA, QDH

6Z9B image
Human Ecto-5'-Nucleotidase (Cd73) In Complex With Aopcp Derivative A830 (Compound 16 In Publication) In The Closed Form (Crystal Form Iii)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.17 Å Release Date: 2020-07-22
Classification: HYDROLASE
Ligands: ZN, CA, QCQ

6XUE image
Human Ecto-5'-Nucleotidase (Cd73) In Complex With A2396 (Compound 74 In Publication) In The Closed Form In Crystal Form Iv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.94 Å Release Date: 2020-04-22
Classification: HYDROLASE
Ligands: ZN, CA, PO4, O1H

6XUG image
Human Ecto-5'-Nucleotidase (Cd73) In Complex With A2410 (Compound 53 In Publication) In The Closed Form In Crystal Form Iv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.09 Å Release Date: 2020-04-22
Classification: HYDROLASE
Ligands: ZN, CA, PO4, O1Q

6XUQ image
Human Ecto-5'-Nucleotidase (Cd73) In Complex With A1618 (Compound 1B In Publication) In The Closed State In Crystal Form Iii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.97 Å Release Date: 2020-04-22
Classification: HYDROLASE
Ligands: ZN, CA, O1T

5HRN image
Hiv Integrase Catalytic Domain Containing F185K Mutation Complexed With Gsk0002
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Resolution:1.75 Å Release Date: 2016-12-14
Classification: TRANSFERASE/INHIBITOR
Ligands: CAC, SO4, EDO, 65P

5HRP image
Hiv Integrase Catalytic Domain Containing F185K + A124T Mutations Complexed With Gsk0002
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Resolution:1.81 Å Release Date: 2016-12-14
Classification: TRANSFERASE/INHIBITOR
Ligands: CAC, SO4, EDO, 65P

5HRR image
Hiv Integrase Catalytic Domain Containing F185K + A124N + T125S Mutations Complexed With Gsk0002
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Resolution:1.88 Å Release Date: 2016-12-14
Classification: TRANSFERASE/INHIBITOR
Ligands: CAC, SO4, EDO, 65P

5HRS image
Hiv Integrase Catalytic Domain Containing F185K + A124N + T125A Mutations Complexed With Gsk0002
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Resolution:1.86 Å Release Date: 2016-12-14
Classification: TRANSFERASE/INHIBITOR
Ligands: CAC, SO4, EDO, 65P

4OJR image
Crystal Structure Of The Hiv-1 Integrase Catalytic Domain With Gsk1264
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Resolution:1.82 Å Release Date: 2014-06-11
Classification: VIRAL PROTEIN
Ligands: 2SQ, CAC, SO4

4BBE image
Aminoalkylpyrimidine Inhibitor Complexes With Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2012-11-21
Classification: TRANSFERASE
Ligands: 3O4

4BBF image
Aminoalkylpyrimidine Inhibitor Complexes With Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2012-11-21
Classification: TRANSFERASE
Ligands: O19

3RJM image
Caspase2 In Complex With Chdi Ligand 33C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.55 Å Release Date: 2011-09-21
Classification: HYDROLASE/HYDROLASE INHIBITOR
Protein Functional Filters:
Feedback Form
Name
Email
Institute
Feedback