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Search Count: 7

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3T8M image
Rational Design Of Pi3K-Alpha Inhibitors That Exhibit Selectivity Over The Pi3K-Beta Isoform

3NZS image
Structure-Based Optimization Of Pyrazolo -Pyrimidine And -Pyridine Inhibitors Of Pi3-Kinase

3NZU image
Structure-Based Optimization Of Pyrazolo -Pyrimidine And -Pyridine Inhibitors Of Pi3-Kinase

3L13 image
Crystal Structures Of Pan-Pi3-Kinase And Dual Pan-Pi3-Kinase/Mtor Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.00 Å Release Date: 2010-02-16
Classification: TRANSFERASE
Ligands: JZW

3L16 image
Discovery Of (Thienopyrimidin-2-Yl)Aminopyrimidines As Potent, Selective, And Orally Available Pan-Pi3-Kinase And Dual Pan-Pi3-Kinase/Mtor Inhibitors For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.90 Å Release Date: 2010-02-16
Classification: TRANSFERASE
Ligands: JZX

3L17 image
Discovery Of (Thienopyrimidin-2-Yl)Aminopyrimidines As Potent, Selective, And Orally Available Pan-Pi3-Kinase And Dual Pan-Pi3-Kinase/Mtor Inhibitors For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.00 Å Release Date: 2010-02-16
Classification: TRANSFERASE
Ligands: JZY

3DBS image
Structure Of Pi3K Gamma In Complex With Gdc0941
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2008-06-17
Classification: TRANSFERASE
Ligands: GD9
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