Search Count: 9
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Crystal Structure Of Nedd4 Hect Domain In Complex With Norclomipramine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2025-06-04 Classification: LIGASE Ligands: EDO, A1ITH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-04
Ligands: EDO, A1ITH
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Crystal Structure Of Nedd4 Hect Domain In Complex With Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2025-06-04 Classification: LIGASE Ligands: A1ITT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-04
Ligands: A1ITT
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Structure Of The Kdm1A/Corest Complex With The Inhibitor 2-[3-{4-Chloro-3-[(4-Chlorophenyl)Ethynyl]Phenyl}-1-(3-Morpholin-4-Ylpropyl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl]-2-Oxoethanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.11 Å Release Date: 2020-06-03 Classification: OXIDOREDUCTASE Ligands: N4K, FAD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-03
Ligands: N4K, FAD, GOL
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Thieno[3,2-B]Pyrrole-5-Carboxamides As Novel Reversible Inhibitors Of Histone Lysine Demethylase Kdm1A/Lsd1: Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, 6W0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, 6W0
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Thieno[3,2-B]Pyrrole-5-Carboxamides As Novel Reversible Inhibitors Of Histone Lysine Demethylase Kdm1A/Lsd1: Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, 6W3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, 6W3
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Thieno[3,2-B]Pyrrole-5-Carboxamides As Novel Reversible Inhibitors Of Histone Lysine Demethylase Kdm1A/Lsd1: Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, 6W1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, 6W1
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Structure Of The Kdm1A/Corest Complex With The Inhibitor 4-Methyl-N-[4-[[4-(1-Methylpiperidin-4-Yl)Oxyphenoxy]Methyl]Phenyl]Thieno[3,2-B]Pyrrole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.34 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, GOL, 6X3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, GOL, 6X3
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Structure Of The Kdm1A/Corest Complex With The Inhibitor 4-Ethyl-N-[3-(Methoxymethyl)-2-[[4-[[(3R)-Pyrrolidin-3-Yl]Methoxy]Phenoxy]Methyl]Phenyl]Thieno[3,2-B]Pyrrole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, GOL, 6X0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, GOL, 6X0
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Structure Of The Kdm1A/Corest Complex With The Inhibitor N-[3-(Ethoxymethyl)-2-[[4-[[(3R)-Pyrrolidin-3-Yl]Methoxy]Phenoxy]Methyl]Phenyl]-4-Methylthieno[3,2-B]Pyrrole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, 6X5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, 6X5, GOL
