Search Count: 35
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Structure Of Ptp1B Complexed With Difluoromethylphosphonate Inhibitor Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2026-05-27 Classification: HYDROLASE/INHIBITOR Ligands: A1C3A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-27
Ligands: A1C3A
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Structure Of Ptp1B Complexed With Difluoromethylphosphonate Inhibitor Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2026-05-27 Classification: HYDROLASE/INHIBITOR Ligands: A1C3B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-27
Ligands: A1C3B
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Structure Of Ptp1B Complexed With Difluoromethylphosphonate Inhibitor Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2026-05-27 Classification: HYDROLASE/INHIBITOR Ligands: A1C3C, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-27
Ligands: A1C3C, DMS
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Structure Of Ptp1B Complexed With Difluoromethylphosphonate Inhibitor Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2026-05-27 Classification: HYDROLASE/INHIBITOR Ligands: A1C3D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-27
Ligands: A1C3D
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Pi3Ka H1047R Co-Crystal Structure With Inhibitor In Cryptic Pocket Near H1047R (Compound 4).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.58 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: YO4, YNZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: YO4, YNZ
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Pi3Ka H1047R Co-Crystal Structure With Inhibitor In Cryptic Pocket (Compound 5).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: YOR, YNZ, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: YOR, YNZ, CL
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Pi3Ka H1047R Co-Crystal Structure With Inhibitors In Two Cryptic Pockets (Compounds 4 And 5).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.35 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: YO4, YOR, YNZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: YO4, YOR, YNZ
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Pi3Ka H1047R Co-Crystal Structure With Inhibitor In Cryptic Pocket Near H1047R (Compound 12).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: 1LT, YQB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: 1LT, YQB
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Pi3Ka H1047R Co-Crystal Structure With Inhibitor In Cryptic Pocket Near H1047R (Compound 7).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: YQ2, 1LT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: YQ2, 1LT
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Prmt5/Mep50 Crystal Structure With Mta And An Achiral, Class 1, Non-Atropisomeric Inhibitor Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2022-08-17 Classification: TRANSFERASE Ligands: NXF, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-17
Ligands: NXF, MTA
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Prmt5/Mep50 Crystal Structure With Sinefungin Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2022-03-16 Classification: TRANSFERASE/INHIBITOR Ligands: SFG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-16
Ligands: SFG
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Kras G12D (Gppcp) With Mrtx-1133
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2022-03-16 Classification: HYDROLASE/INHIBITOR Ligands: 6IC, GCP, GDP, GOL, ACT, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-16
Ligands: 6IC, GCP, GDP, GOL, ACT, MG
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Prmt5/Mep50 Crystal Structure With Mta And Phthalazinone Fragment Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2022-01-26 Classification: TRANSFERASE Ligands: CL, NA, EDO, 81X, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: CL, NA, EDO, 81X, MTA
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Prmt5/Mep50 Crystal Structure With Mta And A Phthalazinone Inhibitor Bound (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: MTA, 84W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: MTA, 84W
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Prmt5/Mep50 Crystal Structure With Mta And A Phthalazinone Inhibitor Bound (Compound (M)-31)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: MTA, 85E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: MTA, 85E
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Prmt5/Mep50 Crystal Structure With Mta And Mrtx-1719 Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: MTA, 85K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: MTA, 85K
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Prmt5/Mep50 With Compound 30 Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: 97L, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: 97L, MTA
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Prmt5/Mep50 With Compound 29 Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: 97X, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: 97X, MTA
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Structure Of Human Anaplastic Lymphoma Kinase In Complex With 2-[(1R)-1-{[2-Amino-5-(1,3-Dimethyl-1H-Pyrazol-4-Yl)Pyridin-3-Yl]Oxy}Ethyl]-4-Fluoro-N,N-Dimethylbenzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2016-08-17 Classification: Transferase/Transferase Inhibitor Ligands: 6YL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-17
Ligands: 6YL
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Structure Of Human Ros1 Kinase Domain In Complex With Pf-06463922
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-03-11 Classification: TRANSFERASE Ligands: 5P8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-11
Ligands: 5P8