Search Count: 37
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Crystal Structure Of Bcl-Xl In Complex With A Benzothiazole-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2021-06-23 Classification: APOPTOSIS Ligands: XZM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-23
Ligands: XZM
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Crystal Structure Of Bcl-2 In Complex With Prodrug Abbv-167
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2021-04-14 Classification: APOPTOSIS Ligands: XZD |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
Ligands: XZD
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Crystal Structure Of Bcl-Xl In Complex With Tetrahydroisoquinoline-Pyridine Based Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-10-21 Classification: APOPTOSIS/APOPTOSIS INHIBITOR Ligands: RQ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-21
Ligands: RQ7
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Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2017-10-04 Classification: signaling protein/inhibitor Ligands: CJY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: CJY
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Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-10-04 Classification: signaling protein/inhibitor Ligands: CN7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: CN7
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Brd4_Bd2-A-35165
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2017-06-28 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 89J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 89J
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Brd4_Bd2_A-1107604
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 0S6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 0S6
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Brd2 Bromodomain2 With A-1360579
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 87D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 87D
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Brd4_Bd2_A-1497627
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 89D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 89D
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Brd4_Bd2_A-1412838
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 88M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 88M
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Brd4_Bd2_A-1342843
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 89G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 89G
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Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2017-05-03 Classification: signaling protein/inhibitor Ligands: 9EA, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-03
Ligands: 9EA, ZN
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Discovery Of A Potent And Selective Bcl-Xl Inhibitor That Demonstrates Thrombocytopenia And Inhibits Tumor Growth In Vivo
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-07-22 Classification: APOPTOSIS/INHIBITOR Ligands: 3CQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-22
Ligands: 3CQ
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Bcl-Xl In Complex With Inhibitor (Compound 10)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-10-15 Classification: APOPTOSIS Ligands: 38H, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-15
Ligands: 38H, EDO, ACT
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Bcl_2-Navitoclax Analog (With Indole) Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2014-01-29 Classification: APOPTOSIS REGULATOR/INHIBITOR Ligands: 1Y1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-29
Ligands: 1Y1
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Bcl_2-Navitoclax (Abt-263) Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2013-08-14 Classification: APOPTOSIS REGULATOR/INHIBITOR Ligands: 1XJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: 1XJ
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Bcl_2-Navitoclax Analog (Without Thiophenyl) Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-08-14 Classification: APOPTOSIS REGULATOR/INHIBITOR Ligands: 1XV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: 1XV
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Crystal Structure Of Hsp90 With N-Aryl-Benzimidazolone I
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-09-21 Classification: CHAPERONE Ligands: MEX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-09-21
Ligands: MEX
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Crystal Structure Of Hsp90 With Ver-49009
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2011-09-21 Classification: CHAPERONE Ligands: BSM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-09-21
Ligands: BSM
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Crystal Structure Of Hsp90 With N-Aryl-Benzimidazolone Ii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2011-09-21 Classification: CHAPERONE Ligands: MEY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-09-21
Ligands: MEY
