Search Count: 8
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Crystal Structure Of C-Terminal Domain Of Msk1 In Complex With In Covalently Bound Literature Rsk2 Inhibitor Pyrrolopyrimidine Cyanoacrylamide Compound 25 (Co-Crystal)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2022-08-31 Classification: TRANSFERASE Ligands: SUU, OXM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-31
Ligands: SUU, OXM
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Crystal Structure Of C-Terminal Domain Of Msk1 In Complex With Covalently Bound With Literature Rsk2 Inhibitor Indazole Cyanoacrylamide Compound 26 (Soak)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2022-07-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1LE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
Ligands: 1LE
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Crystal Structure Of C-Terminal Domain Of Msk1 In Complex With Covalently Bound Pyrrolopyrimidine Compound 20 (Co-Crystal)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2022-07-06 Classification: TRANSFERASE Ligands: O1K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: O1K
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Crystal Structure Of C-Terminal Domain Of Msk1 In Complex With Covalently Bound Pyrrolopyrimidine Compound 23 (Co-Crystal)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2022-07-06 Classification: TRANSFERASE Ligands: O1R, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: O1R, IOD
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Crystal Structure Of C-Terminal Domain Of Msk1 In Complex With Covalently Bound Pyrrolopyrimidine Compound 27 (Co-Crystal)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2022-07-06 Classification: TRANSFERASE Ligands: O10 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: O10
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Identification Of Low Micromolar Sars-Cov-2 Mpro Inhibitors From Hits Identified By In Silico Screens
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2022-05-04 Classification: HYDROLASE Ligands: 4N0 |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: 4N0
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Crystal Structure Of Human Complement C5 In Complex With The K92 Bovine Knob Domain Peptide.
Organism: Bos taurus, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2021-03-10 Classification: IMMUNE SYSTEM Ligands: EDO, CYS, TRS |
Organism: Bos taurus, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-10
Ligands: EDO, CYS, TRS
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Crystal Structure Of Human Complement C5 In Complex With The K8 Bovine Knob Domain Peptide.
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-03-10 Classification: IMMUNE SYSTEM Ligands: EOH, MHA, MPD, CYS, TAM |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2021-03-10
Ligands: EOH, MHA, MPD, CYS, TAM
