Search Count: 26
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Pde2 In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2018-09-19 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, EDO, FKV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: ZN, MG, EDO, FKV
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Pde2 In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2018-09-19 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, FKJ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: ZN, MG, FKJ, EDO
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Pde2 In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2018-09-19 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, FKG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: ZN, MG, FKG, EDO
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Crystal Structure Of Hiv Protease Complexed With (S)-N-(3-Fluoro-2-(2-(1-(Phenylsulfonyl)Piperazin-2-Yl)Ethyl)Phenyl)-3,3-Bis(4-Fluorophenyl)Propanamide
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2018-01-03 Classification: VIRAL PROTEIN/INHIBITOR Ligands: CL, CKD |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2018-01-03
Ligands: CL, CKD
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Crystal Structure Of Hiv Protease Complexed With N-(3-Fluoro-2-(2-((2S,6R)-6-Methyl-1-(Phenylsulfonyl)Piperazin-2-Yl)Ethyl)Phenyl)-3,3-Bis(4-Fluorophenyl)Propanamide
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2018-01-03 Classification: VIRAL PROTEIN/INHIBITOR Ligands: CL, CKM |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2018-01-03
Ligands: CL, CKM
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Crystal Structure Of Hiv Protease Complexed With N-(3-Fluoro-2-(2-((2S,6R)-6-Methyl-1-(Phenylsulfonyl)Piperazin-2-Yl)Ethyl)Phenyl)-3,3-Bis(4-Fluorophenyl)Propanamide
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-01-03 Classification: VIRAL PROTEIN/INHIBITOR Ligands: CL, CKS |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2018-01-03
Ligands: CL, CKS
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Crystal Structure Of Hiv Protease Complexed With N-(3-Fluoro-2-(2-((2S,5S)-5-Methyl-1-(Phenylsulfonyl)Piperazin-2-Yl)Ethyl)Phenyl)-3,3-Bis(4-Fluorophenyl)Propanamide
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2018-01-03 Classification: VIRAL PROTEIN/INHIBITOR Ligands: CL, CKV |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2018-01-03
Ligands: CL, CKV
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Crystal Structure Of Hiv Protease Complexed With N-(3-Fluoro-2-(2-((2S,6S)-6-Methyl-1-(Phenylsulfonyl)Piperazin-2-Yl)Ethyl)Phenyl)-3,3-Bis(4-Fluorophenyl)Propanamide
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2018-01-03 Classification: VIRAL PROTEIN/INHIBITOR Ligands: CL, CKY |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2018-01-03
Ligands: CL, CKY
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Crystal Structure Of Hiv Protease Complexed With N-(2-(2-((6R,9S)-2,2-Dioxido-2-Thia-1,7-Diazabicyclo[4.3.1]Decan-9-Yl)Ethyl)-3-Fluorophenyl)-3,3-Bis(4-Fluorophenyl)Propanamide
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2018-01-03 Classification: VIRAL PROTEIN/INHIBITOR Ligands: CN4, CL |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2018-01-03
Ligands: CN4, CL
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Discovery Of Pyrazolo[1,5A]Pyrimidine-Based Pim1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-09-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 26K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: 26K
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Discovery Of Pyrazolo[1,5A]Pyrimidine-Based Pim1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-09-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 26L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: 26L
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X-Ray Crystal Structure Of Compound 22K Bound To Human Chk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2010-11-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 22K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: 22K
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X-Ray Crystal Structure Of Compound 17R Bound To Human Chk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2010-11-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MI5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: MI5, GOL
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SC8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SC8
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SC9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SC9
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SCE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SCE
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.28 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SCF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SCF
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SCJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SCJ
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SCQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SCQ
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SCW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SCW
