Search Count: 14
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Crystal Structure Of Erk2 In Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2016-07-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6QB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 6QB, EDO
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Crystal Structure Of Cdk2 In Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-07-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6QB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 6QB
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Bcl-Xl In Complex With Inhibitor (Compound 10)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-10-15 Classification: APOPTOSIS Ligands: 38H, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-15
Ligands: 38H, EDO, ACT
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Discovery Of 5,6,7,8-Tetrahydropyrido[3,4-D]Pyrimidine Inhibitors Of Erk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2014-05-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2SH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-21
Ligands: 2SH
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Discovery Of Thiazolobenzoxepin Pi3-Kinase Inhibitors That Spare The Pi3-Kinase Beta Isoform
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-08-28 Classification: Transferase/Transferase Inhibitor Ligands: 1JV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-28
Ligands: 1JV
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X-Ray Crystal Structure Of The Nuclear Hormone Receptor Ppar-Gamma In A Complex With A Compound With Dual Ppar Gamma Agonism And Angiotensin Ii Type I Receptor Antagonism Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2012-03-14 Classification: NUCLEAR PROTEIN Ligands: HIG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-14
Ligands: HIG
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Crystal Structure Of Fxa In Complex With 4,4-Disubstituted Pyrrolidine-1,2-Dicarboxamide Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-04-07 Classification: HYDROLASE Ligands: CA, L1C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-04-07
Ligands: CA, L1C
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Crystal Structure Of Fxa In Complex With 4,4-Disubstituted Pyrrolidine-1,2-Dicarboxamide Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2009-04-07 Classification: HYDROLASE Ligands: L1D, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-04-07
Ligands: L1D, CA
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An Orally Efficacious Factor Xa Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-03-25 Classification: BLOOD CLOTTING Ligands: CA, 230 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-25
Ligands: CA, 230
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Factor Xa Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2007-08-14 Classification: BLOOD CLOTTING Ligands: CA, 237 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-08-14
Ligands: CA, 237
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Crystal Structure Of Factor Vii.Stf Complexed With Pd0297121
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2006-10-18 Classification: HYDROLASE Ligands: CA, GIL, GLC, FUC, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-10-18
Ligands: CA, GIL, GLC, FUC, NAG
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Crystal Structure Of A Ternary Complex Of Factor Viia/Tissue Factor And 2-[[6-[3-(Aminoiminomethyl)Phenoxy]-3,5-Difluro-4-[(1-Methyl-3-Phenylpropyl)Amino]-2-Pyridinyl]Oxy]-Benzoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2006-08-01 Classification: HYDROLASE Ligands: CA, CAC, 03R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-01
Ligands: CA, CAC, 03R
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X-Ray Structure Of The Human Mitogen-Activated Protein Kinase Kinase 2 (Mek2)In A Complex With Ligand And Mgatp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2004-11-23 Classification: TRANSFERASE Ligands: MG, ATP, 5EA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-11-23
Ligands: MG, ATP, 5EA
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X-Ray Structure Of The Human Mitogen-Activated Protein Kinase Kinase 1 (Mek1) In A Complex With Ligand And Mgatp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2004-11-23 Classification: TRANSFERASE Ligands: MG, ATP, BBM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-11-23
Ligands: MG, ATP, BBM
