Search Count: 16
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Human Pi4Kiiib In Complex With Covalently Bound Inhibitor (Compound 4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2023-12-13 Classification: TRANSFERASE Ligands: KHR, MG, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-13
Ligands: KHR, MG, EDO, GOL
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Human Pi4Kiiib In Complex With Covalently Bound Inhibitor (Compound 8)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2023-12-13 Classification: TRANSFERASE Ligands: KIH, MG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-13
Ligands: KIH, MG, EDO
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Human Pi4Kiiib In Complex With Covalently Bound Inhibitor (Compound 11)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2023-12-13 Classification: TRANSFERASE Ligands: MG, KI7, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-13
Ligands: MG, KI7, EDO
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Pi3 Kinase Delta In Complex With 5-[3,6-Dihydro-2H-Pyran-4-Yl]-2-Methoxy-N-[2-Methylpyridin-4-Yl]Pyridine-3-Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-09-29 Classification: SIGNALING PROTEIN Ligands: 7VT |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: 7VT
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Pi3 Kinase Delta In Complex With N-[2-(2-Fluoro-4-{[4-(Propan-2-Yl)Piperazin-1-Yl]Methyl}Phenyl)Pyridin-4-Yl]-2-Methoxy-5-(Morpholin-4-Yl)Pyridine-3-Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2021-09-29 Classification: SIGNALING PROTEIN Ligands: 7XH |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: 7XH
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Pi3 Kinase Delta In Complex With 5-(3,6-Dihydro-2H-Pyran-4-Yl)-2-Methoxy-N-(5-{3-[4-(Propan-2-Yl)Piperazin-1-Yl]Prop-1-Yn-1-Yl}Pyridin-3-Yl)Pyridine-3-Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-09-29 Classification: SIGNALING PROTEIN Ligands: 7XN |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: 7XN
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Pi3 Kinase Delta In Complex With N-[5-(3,6-Dihydro-2H-Pyran-4-Yl)-2-Methoxypyridin-3-Yl]Benzenesulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2021-09-29 Classification: SIGNALING PROTEIN Ligands: 7XW |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: 7XW
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Pi3K Delta In Complex With N[5(7{2[4(2Hydroxypropan2Yl)Piperidin1 Yl]Ethoxy}1,3Dihydro2Benzofuran5Yl)2 Methoxypyridin3Yl]Methanesulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-01-01 Classification: TRANSFERASE Ligands: NQ2 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NQ2
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Pi3K Delta In Complex With 2Methoxyn[2Methoxy5(7{[(2R)4(Oxetan3 Yl)Morpholin2Yl]Methoxy}1,3Dihydro2 Benzofuran5Yl)Pyridin3Yl]Ethane1 Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2020-01-01 Classification: TRANSFERASE Ligands: NQ5 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NQ5
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Pi3K Delta In Complex With N(2Chloro5Phenylpyridin3Yl)Benzenesulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2018-12-26 Classification: TRANSFERASE Ligands: HKQ |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: HKQ
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Pi3K Delta In Complex With N[2Chloro5(3,6Dihydro2Hpyran4Yl)Pyridin3Yl]Methanesulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2018-12-26 Classification: TRANSFERASE Ligands: HKK |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: HKK
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Pi3K Delta In Complex With 1Benzyln[5(3,6Dihydro2Hpyran4Yl)2Methoxypyridin3Yl]2Methyl1Himidazole4Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2018-12-26 Classification: TRANSFERASE Ligands: HKN |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: HKN
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Crystal Structure Of Human Lipoprotein-Associated Phospholipase A2 In Complex With A [1.1.1]Bicyclopentane-Containing Inhibitor At 1.91A Resolution.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2017-02-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CL, 71H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-01
Ligands: CL, 71H
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Crystal Structure Of Mouse Pi3 Kinase Delta In Complex With Gsk2269557
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2015-09-16 Classification: TRANSFERASE Ligands: VVX |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2015-09-16
Ligands: VVX
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Crystal Structure Of Mouse Pi3 Kinase Delta In Complex With Gsk2292767
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2015-09-16 Classification: TRANSFERASE Ligands: OKO |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2015-09-16
Ligands: OKO
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Crystal Structure Of P38 Kinase In Complex With A Pyrrole-2-Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2010-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1GK, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-07
Ligands: 1GK, GOL
