Search Count: 16
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Il17A Homodimer Complexed To Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCE
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Il17A Complexed To Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCW, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCW, CL
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Novel Modes Of Inhibition Of Wild-Type Idh1: Direct Covalent Modification Of His315 With Cmpd1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2018-07-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: CA, ICT, DWP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: CA, ICT, DWP
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Novel Binding Modes Of Inhibition Of Wild-Type Idh1: Allosteric Inhibition With Cmpd2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2018-07-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: LMR, MG, K32 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: LMR, MG, K32
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Novel Modes Of Inhibition Of Wild-Type Idh1: Non-Equivalent Allosteric Inhibition With Cmpd3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2018-07-25 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, DWM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: NAP, DWM
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Novel Modes Of Inhibition Of Wild-Type Idh1:Direct Covalent Modification Of His315 With Cmpd11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2018-07-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: MG, ICT, DWJ, NAP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: MG, ICT, DWJ, NAP
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Novel Modes Of Inhibition Of Wild-Type Idh1: Direct Covalent Modification Of His315 With Cmpd13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2018-07-25 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: ICT, DWG, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: ICT, DWG, CA
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Novel Modes Of Inhibition Of Wild-Type Idh1: Direct Covalent Modification Of His315 With Cmpd15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2018-07-25 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: CA, ICT, DWS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: CA, ICT, DWS
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The Dodecameric Human Ruvbl1:Ruvbl2 Complex With Truncated Domains Ii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2011-10-05 Classification: HYDROLASE Ligands: ATP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: ATP
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Crystal Structure Of Wild-Type Plk-1 Kinase Domain In Complex With A Selective Darpin
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-04-01 Classification: TRANSFERASE |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2008-04-01
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3D Structure Of The Human Ruvb-Like Helicase Ruvbl1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2006-10-23 Classification: HYDROLASE Ligands: ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-10-23
Ligands: ADP
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Structural Basis For The Glucocorticoid Response In A Mutant Human Androgen Receptor (Arccr) Derived From An Androgen-Independent Prostate Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2003-01-16 Classification: ANDROGEN RECEPTOR Ligands: ZK5, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-01-16
Ligands: ZK5, PO4
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Human Androgen Receptor Ligand Binding In Complex With The Ligand Metribolone (R1881)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2001-06-14 Classification: ANDROGEN RECEPTOR Ligands: R18 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2001-06-14
Ligands: R18
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Human Progesteron Receptor Ligand Binding Domain In Complex With The Ligand Metribolone (R1881)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2001-06-14 Classification: HUMAN PROGESTERONE RECEPTOR Ligands: R18 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2001-06-14
Ligands: R18
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Catalytic Domain Of Vampire Bat (Desmodus Rotundus) Saliva Plasminogen Activator In Complex With Egr-Cmk (Glu-Gly-Arg Chloromethyl Ketone)
Organism: Desmodus rotundus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 1999-03-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0GJ |
Organism: Desmodus rotundus
Method: X-RAY DIFFRACTION
Release Date: 1999-03-23
Ligands: 0GJ
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Thrombin Inhibitor From Triatoma Pallidipennis
Organism: Triatoma pallidipennis, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 1998-12-30 Classification: COMPLEX (BLOOD COAGULATION/INHIBITOR) |
Organism: Triatoma pallidipennis, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 1998-12-30
