Search Count: 6
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Discovery Of A Small Molecule Itk And Pan-Trk Kinase Inhibitor (Pf-07245303) For The Potential Topical Treatment Of Atopic Dermatitis
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2025-11-19 Classification: SIGNALING PROTEIN Ligands: A1B66 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-19
Ligands: A1B66
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Crystal Structure Of Human Set And Mynd Domain Containing Protein 2 With Mtf9975
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2018-03-14 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, EW4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: ZN, EW4
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Selective Pharmacological Inhibition Of The Creb Binding Protein Bromodomain Regulates Inflammatory Cytokines In Macrophages And Rgs4 In Neurons
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2016-04-20 Classification: TRANSCRIPTION/INHIBITOR Ligands: 53W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 53W
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Selective Pharmacological Inhibition Of The Creb Binding Protein Bromodomain Regulates Inflammatory Cytokines In Macrophages And Rgs4 In Neurons
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2016-04-20 Classification: TRANSCRIPTION/INHIBITOR Ligands: 53W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 53W
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Bromo Domain Of Creb Binding Protein
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3OT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 3OT
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Direct Photocapture Of Bromodomains Using Tropolone Chemical Probes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2015-10-28 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 3OT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 3OT, EDO
