Search Count: 37
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Crystal Structure Of Human Pi3Ka (P110A Subunit) With Mmv085400 Bound To The Active Site Determined At 2.9 Angstroms Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2022-05-04 Classification: TRANSFERASE/INHIBITOR Ligands: ZHY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: ZHY
 |
Prmt5:Mep50 Complexed With Inhibitor Pf-06939999
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ZR1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR1
 |
Prmt5:Mep50 Complexed With Inhibitor Pf-06855800
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2021-11-17 Classification: Transferase/Transcription Ligands: ZR4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR4
 |
Prmt5:Mep50 Complexed With Adenosine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ADN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ADN
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Prmt5(M420T Mutant):Mep50 Complexed With Inhibitor Pf-06855800
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ZR4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR4
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Prmt5(M420T Mutant):Mep50 Complexed With Inhibitor Pf-06939999
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2021-11-17 Classification: transferase/Transcription Ligands: ZR1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR1
 |
Crystal Structure Of Pi3Kalpha Selective Inhibitor Pf-06843195
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VXY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VXY
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Crystal Structure Of Pi3Kalpha Selective Inhibitor 11-1575
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VY4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VY4
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Crystal Structure Of Pi3Kalpha Inhibitor 10-5429
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VY1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VY1
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Crystal Structure Of Pi3Kalpha Inhibitor 4-0686
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VYP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VYP
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Crystal Structure Of Human Naa50 In Complex With A Cofactor Derived Inhibitor (Compound 1)
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: COA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: COA
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Crystal Structure Of Human Naa50 In Complex With A Truncated Cofactor Derived Inhibitor (Compound 2)
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: U44 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: U44
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Crystal Structure Of Human Naa50 In Complex With An Inhibitor (Compound 3) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: COA, U3V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: COA, U3V
 |
Crystal Structure Of Human Naa50 In Complex With Coa And An Inhibitor (Compound 4A) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2020-07-01 Classification: TRANSFERASE Ligands: COA, U2J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: COA, U2J
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Crystal Structure Of Human Naa50 In Complex With Accoa And An Inhibitor (Compound 4A) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.07 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: ACO, U2J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: ACO, U2J
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Crystal Structure Of Human Naa50 In Complex With Accoa And An Inhibitor (Compound 4B) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: ACO, U3Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: ACO, U3Y
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Structure Of Hs/Acprc2 In Complex With 5,8-Dichloro-2-[(4-Methoxy-6-Methyl-2-Oxo-1,2-Dihydropyridin-3-Yl)Methyl]-7-[(R)-Methoxy(Oxetan-3-Yl)Methyl]-3,4-Dihydroisoquinolin-1(2H)-One
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2017-12-27 Classification: Transferase/Transferase Inhibitor Ligands: ZN, CJD |
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: ZN, CJD
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Structure Of Hs/Acprc2 In Complex With 5,8-Dichloro-7-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-2-[(4,6-Dimethyl-2-Oxo-1,2-Dihydropyridin-3-Yl)Methyl]-3,4-Dihydroisoquinolin-1(2H)-One
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2017-12-27 Classification: METAL BINDING PROTEIN Ligands: ZN, CJG |
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: ZN, CJG
 |
Structure Of Human Anaplastic Lymphoma Kinase In Complex With 2-[(1R)-1-{[2-Amino-5-(1,3-Dimethyl-1H-Pyrazol-4-Yl)Pyridin-3-Yl]Oxy}Ethyl]-4-Fluoro-N,N-Dimethylbenzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2016-08-17 Classification: Transferase/Transferase Inhibitor Ligands: 6YL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-17
Ligands: 6YL
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Structure Of Hs/Acprc2 In Complex With A Pyridone Inhibitor
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2016-05-04 Classification: transferase/transferase inhibitor Ligands: 6BN, ZN |
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 6BN, ZN