Search Count: 13
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Crystal Structure Of Human Folate Receptor Alpha In Complex With Novel Antifolate Agf183
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2016-08-10 Classification: SIGNALING PROTEIN Ligands: 83A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: 83A
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Human Gar Transformylase In Complex With Gar And (4-{[2-(2-Amino-4-Oxo-4,7-Dihydro-3H-Pyrrolo[2,3-D]Pyrimidin-6-Yl)Ethyl]Amino}Benzoyl)-L-Glutamic Acid (Agf183)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-08-10 Classification: ligase/ligase inhibitor Ligands: GAR, 83A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: GAR, 83A
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Human Gar Transformylase In Complex With Gar And N-{4-[4-(2-Amino-4-Oxo-4,7-Dihydro-3H-Pyrrolo[2,3-D]Pyrimidin-6-Yl)Benzyl]Benzoyl}-L-Glutamic Acid (Agf23)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GAR, 3Y9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: GAR, 3Y9
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Human Gar Transformylase In Complex With Gar And N-{4-[4-(2-Amino-4-Oxo-3,4-Dihydrothieno[2,3-D]Pyrimidin-6-Yl)-Butyl]Benzoyl}-L-Glutamic Acid (Agf50)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2016-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GAR, 3YA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: GAR, 3YA
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Human Gar Transformylase In Complex With Gar And N-({5-[(2-Amino-4-Oxo-4,7-Dihydro-3H-Pyrrolo[2,3-D]Pyrimidin-6-Yl)Butyl]Thiophen-2-Yl}Carbonyl)-L-Glutamic Acid (Agf71)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2016-04-20 Classification: transferase/transferase inhibitor Ligands: GAR, G71 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: GAR, G71
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Human Gar Transformylase In Complex With Gar And N-({5-[(2-Amino-4-Oxo-4,7-Dihydro-3H-Pyrrolo[2,3-D]Pyrimidin-6-Yl)Propyl]Thiophen-2-Yl}Carbonyl)-L-Glutamic Acid (Agf94)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2016-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GAR, G94 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: GAR, G94
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Human Gar Transformylase In Complex With Gar And (S)-2-({4-[4-(2-Amino-4-Oxo-4,7-Dihydro-3H-Pyrrolo[2,3-D]-Pyrimidin-6-Yl)Butyl]Thiophene-2-Carbonyl}Amino)Pentanedioic Acid (Agf117)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2016-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GAR, 3YB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: GAR, 3YB
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Human Gar Transformylase In Complex With Gar And (S)-2-({5-[4-(2-Amino-4-Oxo-4,7-Dihydro-3H-Pyrrolo[2,3-D]-Pyrimidin-6-Yl)Butyl]Thiophene-3-Carbonyl}Amino)Pentanedioic Acid (Agf118)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GAR, 3YC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: GAR, 3YC
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Human Gar Transformylase In Complex With Gar And (S)-2-(7-(2-Amino-4-Oxo-4,7-Dihydro-3H-Pyrrolo[2,3-D]Pyrimidin-6-Yl)Heptanamido)Pentanedioic Acid (Agf145)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GAR, 3YD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: GAR, 3YD
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Human Gar Transformylase In Complex With Gar And (S)-2-(8-(2-Amino-4-Oxo-4,7-Dihydro-3H-Pyrrolo[2,3-D]Pyrimidin-6-Yl)Octanamido)Pentanedioic Acid (Agf147)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2016-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GAR, 3YE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: GAR, 3YE
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Human Gar Transformylase In Complex With Gar And (S)-2-({4-[3-(2-Amino-4-Oxo-4,7-Dihydro-3H-Pyrrolo[2,3-D]Pyrimidin-6-Yl)-Propyl]-Thiophene-2-Carbonyl}-Amino)-Pentanedioic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2015-12-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GAR, 3YF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: GAR, 3YF
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Human Gar Transformylase In Complex With Gar And (S)-2-({5-[3-(2-Amino-4-Oxo-4,7-Dihydro-3H-Pyrrolo[2,3-D]Pyrimidin-6-Yl)-Propyl]-Thiophene-3-Carbonyl}-Amino)-Pentanedioic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2015-12-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GAR, 3YG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: GAR, 3YG
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Human Gar Transformylase In Complex With Gar And Pemetrexed
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-12-16 Classification: transferase/transferase inhibitor Ligands: 4DW, GAR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: 4DW, GAR