Search Count: 13
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Crystal Structure Of Egfr Lrtm With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2022-07-27 Classification: SIGNALING PROTEIN Ligands: GOL, QCR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-27
Ligands: GOL, QCR
 |
Crystal Structure Of Egfr Lrtm With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2022-07-27 Classification: SIGNALING PROTEIN Ligands: GOL, QFO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-27
Ligands: GOL, QFO
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Crystal Structure Of Cdk9-Cyclin T1 Bound By Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2021-10-27 Classification: TRANSFERASE Ligands: UT5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-27
Ligands: UT5
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Cdk9-Cyclin-T1 Complex Bound By Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.37 Å Release Date: 2020-12-23 Classification: TRANSFERASE Ligands: Q6E, TRS, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-23
Ligands: Q6E, TRS, PO4
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A Novel Oral Selective Estrogen Receptor Down-Regulator, Azd9496, Drives Tumour Growth Inhibition In Estrogen Receptor Positive And Esr1 Mutant Models
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2015-12-16 Classification: SIGNALING PROTEIN Ligands: KE9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: KE9
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Optimization Of A Novel Binding Motif To To (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-Fluoro-2-Methylpropyl)-3-Methyl-2,3,4,9-Tetrahydro-1H- Pyrido(3,4-B)Indol-1-Yl)Phenyl)Acrylic Acid (Azd9496), A Potent And Orally Bioavailable Selective Estrogen Receptor Downregulator And Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-10-14 Classification: SIGNALING PROTEIN Ligands: XBR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: XBR
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Optimization Of A Novel Binding Motif To To (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-Fluoro-2-Methylpropyl)-3-Methyl-2,3,4,9-Tetrahydro-1H- Pyrido(3,4-B)Indol-1-Yl)Phenyl)Acrylic Acid (Azd9496), A Potent And Orally Bioavailable Selective Estrogen Receptor Downregulator And Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-10-14 Classification: SIGNALING PROTEIN Ligands: GW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: GW5
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Oxyphenylpropenoic Acids As Oral Selective Estrogen Receptor Down- Regulators.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2015-04-22 Classification: SIGNALING PROTEIN Ligands: 85Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: 85Z
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Mmp13 In Complex With A Reverse Hydroxamate Zn-Binder
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2014-03-05 Classification: HYDROLASE Ligands: ZN, CA, NA, AZ4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-03-05
Ligands: ZN, CA, NA, AZ4
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Mmp13 In Complex With A Piperazine Hydantoin Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-03-05 Classification: HYDROLASE Ligands: ZN, CA, NA, AZ6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-03-05
Ligands: ZN, CA, NA, AZ6
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Mmp13 In Complex With A Novel Selective Non Zinc Binding Inhibitor Cmpd22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-12-21 Classification: HYDROLASE Ligands: 3W5, HAE, GOL, ZN, CA, NA, 3W4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-21
Ligands: 3W5, HAE, GOL, ZN, CA, NA, 3W4
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Adamts1 In Complex With A Novel N-Hydroxyformamide Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-03-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: QGF, ZN, CD, NI, MG, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: QGF, ZN, CD, NI, MG, NA
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Adamts1 In Complex With N-Hydroxyformamide Inhibitors Of Adam-Ts4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2011-03-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CD, NI, MG, NA, QHF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: ZN, CD, NI, MG, NA, QHF