Search Count: 11
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Tryptophan 5-Hydroxylase In Complex With Inhibitor (3~{S})-8-[2-Azanyl-6-[(1~{R})-1-(4-Chloranyl-2-Phenyl-Phenyl)-2,2,2-Tris(Fluoranyl)Ethoxy]Pyrimidin-4-Yl]-2,8-Diazaspiro[4.5]Decane-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-01-25 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: FE, 6Z4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: FE, 6Z4
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Optimization Of Spirocyclic Proline Tryptophanhydroxylase-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2017-01-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: FE, TRS, CCN, 7H5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: FE, TRS, CCN, 7H5
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Discovery Of Acyl Guanidine Tryptophan Hydroxylase-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-05-25 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: FE, TRS, GOL, 6H5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: FE, TRS, GOL, 6H5
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Crystal Structure Of Human Chymase In Complex With Fragment Inhibitor 6-Chloro-1,3-Dihydro-2H-Indol-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-05-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, NAG, ES2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: ZN, NAG, ES2
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Crystal Structure Of Human Chymase In Complex With Fragment Inhibitor 6-Chloro-2,3-Dihydro-1H-Isoindol-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-05-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, ZN, 1P7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: NAG, ZN, 1P7
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Crystal Structure Of Human Chymase In Complex With Fragment 6-Bromo-1,3-Dihydro-2H-Indol-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2013-05-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, ZN, 1P8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: NAG, ZN, 1P8
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Crystal Structure Of Human Chymase In Complex With Fragment Linked Benzimidazolone Inhibitor: (3S)-3-{3-[(6-Bromo-2-Oxo-2,3-Dihydro-1H-Indol-4-Yl)Methyl]-2-Oxo-2,3-Dihydro-1H-Benzimidazol-1-Yl}Hexanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2013-05-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, NAG, 1P9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: ZN, NAG, 1P9
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Crystal Structure Of Human Chymase With Benzimidazolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2011-07-20 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, ZN, 0BB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-07-20
Ligands: NAG, ZN, 0BB
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Crystal Structure Of Soluble Epoxide Hydrolase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.79 Å Release Date: 2010-04-28 Classification: HYDROLASE Ligands: 24D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-04-28
Ligands: 24D
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Crystal Structure Of Soluble Epoxide Hydrolase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2009-10-13 Classification: HYDROLASE Ligands: 33N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-13
Ligands: 33N
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Crystal Structure Of Soluble Epoxide Hydrolase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2009-10-13 Classification: HYDROLASE Ligands: 34N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-13
Ligands: 34N