Search Count: 15
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Egfr (T79M/V948R) In Complex With Naquotinib And An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2022-02-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: VNS, 8RC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: VNS, 8RC
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Egfr L858R/V948R In Complex With Osimertinib And Allosteric Inhibitor Jbj-09-063
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2021-09-15 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: VNS, YY3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VNS, YY3
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Egfr Kinase (L858R/V948R) In Complex With Allosteric Inhibitor Jbj-09-063
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2021-09-15 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: MG, ANP, VNS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: MG, ANP, VNS
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Egfr Kinase (T790M/V948R) In Complex With Pf-06747775
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: 8BS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: 8BS
 |
Egfr Kinase (T790M/V948R) In Complex With Pf-06747775 And Jbj-04-125-02
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ANP, MG, JBJ, 8BS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: ANP, MG, JBJ, 8BS
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Egfr Kinase (T790M/V948R) In Complex With Az5104
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: VO7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: VO7
 |
Egfr Kinase (T790M/V948R) In Complex With Osimertinib And Eai045
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ANP, MG, 9LL, YY3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: ANP, MG, 9LL, YY3
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Egfr Kinase (T790M/V948R) In Complex With Osimertinib And Jbj-04-125-02
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ANP, MG, JBJ, YY3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: ANP, MG, JBJ, YY3
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Egfr Kinase (T790M/V948R) In Complex With Osimertinib And Jbj-09-063
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: YY3, VNS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: YY3, VNS
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Egfr(T790M/V948R) In Complex With Azd9291 And Ddc4002
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2021-06-30 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: Q6K, NQ1, MG, ANP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-30
Ligands: Q6K, NQ1, MG, ANP
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Crystal Structure Of Egfr With Mutant-Selective Dihydrodibenzodiazepinone Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-12-18 Classification: Transferase/Transferase Inhibitor Ligands: NQ1, ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-18
Ligands: NQ1, ANP, MG
 |
Crystal Structure Of Egfr In Complex With Eai045
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2019-12-18 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: MG, ANP, 9LL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-18
Ligands: MG, ANP, 9LL
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Egfr In Complex With A Dihydrodibenzodiazepinone Allosteric Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-12-18 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ANP, O57, MG, AMP, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-18
Ligands: ANP, O57, MG, AMP, EDO
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Egfr With An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-06-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, ANP, JBJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-05
Ligands: MG, ANP, JBJ
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Discovery Of A Highly Potent And Broadly Effective Egfr And Her2 Exon 20 Insertion Mutant Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2018-07-18 Classification: Transferase/Transferase Inhibitor Ligands: FZP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: FZP