Search Count: 61
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Biphenyl-Derived Compound 26 (Mi2456)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1JA6, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1JA6, CA, NA, CL, DMS, NAG
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Biphenyl-Derived Compound 42 (Mi2464)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: CA, NA, CL, DMS, NAG, A1JA1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: CA, NA, CL, DMS, NAG, A1JA1
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Biphenyl-Derived Compound 34 (Mi2470)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: CA, NA, CL, DMS, NAG, A1JA2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: CA, NA, CL, DMS, NAG, A1JA2
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Biphenyl-Derived Compound 27 (Mi2471)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1JA3, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1JA3, CA, NA, CL, DMS, NAG
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Biphenyl-Derived Compound 13 (Mi3102)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: CA, NA, CL, DMS, NAG, A1JA5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: CA, NA, CL, DMS, NAG, A1JA5
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Biphenyl-Derived Compound 24 (Mi3140)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1JA4, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1JA4, CA, NA, CL, DMS, NAG
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High-Resolution X-Ray Structure Of Human Pc1/3 (Pcsk1) Prodomain R77A,R80A,R81A Triple-Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2025-09-10 Classification: HYDROLASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Pc1/3 (Pcsk1) Prodomain Mutant R78K,R80A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2025-09-10 Classification: HYDROLASE Ligands: CA, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: CA, NA
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Pc1/3 (Pcsk1) Prodomain Mutant R77A,R80A,R81A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2025-09-10 Classification: HYDROLASE Ligands: CA, NA, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: CA, NA, NAG
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X-Ray Structure Of Furin (Pcsk3) In Complex With Guanidinomethyl-Phac-Can-Tle-Can-6-(Aminomethyl)-3-Amino-Isoindol
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2024-03-13 Classification: HYDROLASE Ligands: CA, NA, CL, DMS |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2024-03-13
Ligands: CA, NA, CL, DMS
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X-Ray Structure Of Furin (Pcsk3) In Complex With Benzamidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-10-04 Classification: HYDROLASE Ligands: BEN, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-04
Ligands: BEN, CA, NA, CL, DMS, NAG
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X-Ray Structure Of Furin (Pcsk3) In Complex With 1H-Isoindol-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-10-04 Classification: HYDROLASE Ligands: F05, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-04
Ligands: F05, CA, NA, CL, DMS, NAG
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X-Ray Structure Of Furin (Pcsk3) In Complex With Guanidinomethyl-Phac-R-Tle-K-6-(Aminomethyl)-3-Amino-Isoindol
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-10-04 Classification: HYDROLASE Ligands: CA, NA, CL, DMS |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2023-10-04
Ligands: CA, NA, CL, DMS
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X-Ray Structure Of Furin In Complex With The Dichlorophenylpyridine-Based Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2022-04-20 Classification: HYDROLASE Ligands: CA, NA, CL, I1G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-20
Ligands: CA, NA, CL, I1G
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X-Ray Structure Of Furin In Complex With The Dichlorophenylpyridine-Based Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2022-04-20 Classification: HYDROLASE Ligands: I0T, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-20
Ligands: I0T, CA, NA, CL, DMS, NAG
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X-Ray Structure Of Furin In Complex With The Dichlorophenylpyridine-Based Inhibitor 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2022-04-20 Classification: HYDROLASE Ligands: I0W, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-20
Ligands: I0W, CA, NA, CL, DMS, NAG
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X-Ray Structure Of Furin In Complex With The Dichlorophenylpyridine-Based Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2022-04-20 Classification: HYDROLASE Ligands: I0Q, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-20
Ligands: I0Q, CA, NA, CL, DMS, NAG
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X-Ray Structure Of Furin In Complex With The Dichlorophenylpyridine-Based Inhibitor 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-04-13 Classification: HYDROLASE Ligands: CA, NA, CL, I0M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-13
Ligands: CA, NA, CL, I0M
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Crystal Structure Of Human Legumain In Complex With Gly-Ser-Asn Peptide
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2021-09-22 Classification: HYDROLASE Ligands: NAG |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: NAG
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X-Ray Structure Of Furin In Complex With The Guanylhydrazone-Based Inhibitor 1 (Bev241)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2021-09-01 Classification: HYDROLASE Ligands: UYN, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-01
Ligands: UYN, CA, NA, CL, DMS, NAG
