Search Count: 12
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Estrogen Receptor Alpha Ligand Binding Domain Y537S In Complex With 4-Hydroxytamoxifen
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2022-06-15 Classification: TRANSCRIPTION Ligands: OHT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-15
Ligands: OHT
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Raloxifene In Complex With Estrogen Receptor Alpha Ligand Binding Domain Y537S Mutation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2022-06-15 Classification: TRANSCRIPTION Ligands: RAL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-15
Ligands: RAL
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Estrogen Receptor Alpha Ligand Binding Domain In Complex With A Methylated Lasofoxifene Derivative With Selective Estrogen Receptor Degrader Properties
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-06-15 Classification: TRANSCRIPTION Ligands: R3V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-15
Ligands: R3V
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Estrogen Receptor Alpha Ligand Binding Domain In Complex With A Methylated Lasofoxifene Derivative That Increases Receptor Resonance Time In The Nucleus Of Breast Cancer Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-06-15 Classification: TRANSCRIPTION Ligands: RL4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-15
Ligands: RL4
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Estrogen Receptor Alpha Ligand Binding Domain In Complex With Ru39411
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2022-06-15 Classification: TRANSCRIPTION Ligands: QYM, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-15
Ligands: QYM, MG
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Estrogen Receptor Alpha Ligand Binding Domain Y537S Mutant In Complex With A Methylated Lasofoxifene Derivative That Possesses Selective Estrogen Receptor Degrader Activities
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2022-06-15 Classification: TRANSCRIPTION Ligands: R3V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-15
Ligands: R3V
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Estrogen Receptor Alpha Ligand Binding Domain Y537S Mutant In Complex With A Methylated Lasofoxifene Derivative That Enhances Estrogen Receptor Alpha Nuclear Resonance Time
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-06-15 Classification: TRANSCRIPTION Ligands: RL4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-15
Ligands: RL4
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Estrogen Receptor Alpha Ligand Binding Domain Y537S Mutant In Complex With Ru39411
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2022-05-04 Classification: TRANSCRIPTION Ligands: NYU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: NYU
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Estrogen Receptor Alpha Ligand Binding Domain In Complex With Raloxifene
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2020-11-18 Classification: TRANSCRIPTION Ligands: RAL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: RAL
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Estrogen Receptor Alpha Ligand Binding Domain In Complex With The Selective Estrogen Receptor Modulator Clomiphene
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-09-16 Classification: TRANSFERASE Ligands: 53Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: 53Q
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Estrogen Receptor Alpha Ligand Binding Domain Y537S In Complex With Lsz102
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-12-25 Classification: TRANSCRIPTION Ligands: C6V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: C6V
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Bazedoxifene In Complex With Y537S Estrogen Receptor Alpha Ligand Binding Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-11-20 Classification: TRANSCRIPTION Ligands: 29S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-20
Ligands: 29S
