Search Count: 43
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Structure Of Human Sting In Complex With Mk-1454
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2022-04-06 Classification: IMMUNE SYSTEM Ligands: ZEV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-06
Ligands: ZEV
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Sting C-Terminal Domain Complexed With Non-Cyclic Dinucleotide Compound Msa-2
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2020-08-19 Classification: IMMUNE SYSTEM Ligands: QAD |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: QAD
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Sting C-Terminal Domain Complexed With Non-Cyclic Dinucleotide Compound 3
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2020-08-19 Classification: IMMUNE SYSTEM Ligands: QAV |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: QAV
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Sting C-Terminal Domain Complexed With Non-Cyclic Dinucleotide Compound 9
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2020-08-19 Classification: IMMUNE SYSTEM Ligands: QB1 |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: QB1
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Sting C-Terminal Domain Complexed With Non-Cyclic Dinucleotide Compound 10
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2020-08-19 Classification: IMMUNE SYSTEM Ligands: QB7 |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: QB7
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Sting C-Terminal Domain Complexed With Non-Cyclic Dinucleotide Compound 11
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2020-08-19 Classification: IMMUNE SYSTEM Ligands: QBA |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: QBA
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Sting C-Terminal Domain Complexed With Non-Cyclic Dinucleotide Compound 12
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-08-19 Classification: IMMUNE SYSTEM Ligands: QBD |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: QBD
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Sting C-Terminal Domain Complexed With Non-Cyclic Dinucleotide Compound 6
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2020-08-19 Classification: IMMUNE SYSTEM Ligands: QBG |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: QBG
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Sting C-Terminal Domain Complexed With Non-Cyclic Dinucleotide Compound 4
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2020-08-19 Classification: IMMUNE SYSTEM Ligands: QBJ |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: QBJ
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Human Arginase1 Complexed With Bicyclic Inhibitor Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2020-05-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MN, QR1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: MN, QR1
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Human Arginase1 Complexed With Bicyclic Inhibitor Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2020-05-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MN, QR4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: MN, QR4
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Human Arginase1 Complexed With Bicyclic Inhibitor Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2020-05-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MN, QRA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: MN, QRA
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Human Arginase1 Complexed With Bicyclic Inhibitor Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2020-05-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MN, QRJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: MN, QRJ
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Bace1 In Complex With (S)-5-(3-Chloro-5-(5-(Prop-1-Yn-1-Yl)Pyridin-3-Yl)Thiophen-2-Yl)-2,5-Dimethyl-1,2,4-Thiadiazinan-3-Iminium 1,1-Dioxide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 66J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 66J
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Bace1 In Complex With 4-(3-(Furan-2-Carboxamido)Phenyl)-1-Methyl-5-Oxo-4-Phenylimidazolidin-2-Iminium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: TLA, 66H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: TLA, 66H
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Bace1 In Complex With (R)-N-(3-(3-Amino-2,5-Dimethyl-1,1-Dioxido-5,6-Dihydro-2H-1,2,4-Thiadiazin-5-Yl)-4-Fluorophenyl)-5-Fluoropicolinamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 66F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 66F
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Bace-1 In Complex With (7Ar)-7A-(4-(3-Cyanophenyl)Thiophen-2-Yl)-6-(5-Fluoropyrimidin-2-Yl)-3-Methyl-4-Oxooctahydro-2H-Pyrrolo[3,4-D]Pyrimidin-2-Iminium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2016-03-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: TLA, 60Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-16
Ligands: TLA, 60Y
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Bace-1 Incomplex With (7Ar)-7A-(4-(3-Cyanophenyl)Thiophen-2-Yl)-6-(5-Fluoro-4-Methoxypyrimidin-2-Yl)-3-Methyl-4-Oxooctahydro-2H-Pyrrolo[3,4-D]Pyrimidin-2-Iminium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2016-03-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: TLA, 60W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-16
Ligands: TLA, 60W
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Bace-1 Incomplex With (7Ar)-7A-(5-Cyanothiophen-2-Yl)-6-(5-Fluoro-4-Methoxy-6-Methylpyrimidin-2-Yl)-3-Methyl-4-Oxooctahydro-2H-Pyrrolo[3,4-D]Pyrimidin-2-Iminium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2016-03-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 60V, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-16
Ligands: 60V, TLA
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Bace-1 In Complex With (7Ar)-7A-(5-Cyanothiophen-2-Yl)-6-(4-Ethoxy-5-Fluoro-6-Methylpyrimidin-2-Yl)-3-Methyl-4-Oxooctahydro-2H-Pyrrolo[3,4-D]Pyrimidin-2-Iminium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-03-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 60U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-16
Ligands: 60U
