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4JQ7 image
Crystal Structure Of Egfr Kinase Domain In Complex With Compound 2A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.73 Å Release Date: 2013-06-19
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: KJQ

4JQ8 image
Crystal Structure Of Egfr Kinase Domain In Complex With Compound 4B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.83 Å Release Date: 2013-06-19
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: KJ8

4JR3 image
Crystal Structure Of Egfr Kinase Domain In Complex With Compound 3G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2013-06-19
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: KJR

4JRV image
Crystal Structure Of Egfr Kinase Domain In Complex With Compound 4C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2013-06-19
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: KJV

4JBO image
Novel Aurora Kinase Inhibitors Reveal Mechanisms Of Hurp In Nucleation Of Centrosomal And Kinetochore Microtubules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.49 Å Release Date: 2013-06-05
Classification: TRANSFERASE
Ligands: WPH

4JBP image
Novel Aurora Kinase Inhibitors Reveal Mechanisms Of Hurp In Nucleation Of Centrosomal And Kinetochore Microtubules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.45 Å Release Date: 2013-06-05
Classification: TRANSFERASE
Ligands: YPH

4JBQ image
Novel Aurora Kinase Inhibitors Reveal Mechanisms Of Hurp In Nucleation Of Centrosomal And Kinetochore Microtubules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2013-06-05
Classification: TRANSFERASE
Ligands: VX6

3NOA image
Crystal Structure Of Human Ppar-Gamma Ligand Binding Domain Complex With A Potency Improved Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.98 Å Release Date: 2011-06-29
Classification: TRANSCRIPTION
Ligands: 5BC

3M11 image
Crystal Structure Of Aurora A Kinase Complexed With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.75 Å Release Date: 2011-03-09
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: AKI

3K5U image
Identification, Sar Studies And X-Ray Cocrystal Analysis Of A Novel Furano-Pyrimidine Aurora Kinase A Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2010-10-13
Classification: TRANSFERASE
Ligands: PFQ

3GBK image
Crystal Structure Of Human Ppar-Gamma Ligand Binding Domain Complexed With A Potent And Selective Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2009-12-29
Classification: ligand binding protein
Ligands: 2PQ

3FDN image
Structure-Based Drug Design Of Novel Aurora Kinase A Inhibitors: Structure Basis For Potency And Specificity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2009-09-15
Classification: TRANSFERASE
Ligands: MMH
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