Search Count: 14
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Bace1 In Complex With 4-(Cyclohexylamino)-1-(3-Fluorophenyl)-8-(3-Isopropoxybenzyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QA
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Bace1 In Complex With 8-(3-((1-Aminopropan-2-Yl)Oxy)Benzyl)-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-08-05 Classification: Hydrolase/Hydrolase inhibitor Ligands: 4QD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QD
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Bace1 In Complex With 8-Benzyl-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-7-Methyl-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QF
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Hiv Protease Complexed With Compound 10B
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-06-30 Classification: TRANSFERASE Ligands: 595, CL |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2010-06-30
Ligands: 595, CL
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Discovery Of Aminoheterocycles As A Novel Beta-Secretase Inhibitor Class
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2009-07-07 Classification: HYDROLASE Ligands: B35 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-07
Ligands: B35
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Crystal Structure Of Hiv-1 Protease Complexed With Pl-100
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2008-07-22 Classification: HYDROLASE Ligands: A00 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2008-07-22
Ligands: A00
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Crystal Structure Of Human Beta Secretase Complexed With Ixs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2008-04-22 Classification: HYDROLASE Ligands: IXS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-22
Ligands: IXS
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Crystal Structure Of Human Beta-Secretase Complexed With L-L000430,469
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2005-12-06 Classification: HYDROLASE Ligands: 3BN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-12-06
Ligands: 3BN
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Crystal Structure Of Human Beta Secretase Complexed With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2005-10-18 Classification: HYDROLASE Ligands: 5HA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-10-18
Ligands: 5HA
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Thrombin In Complex With An Oxazolopyridine Inhibitor 21
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2005-09-27 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 382 |
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-09-27
Ligands: 382
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Thrombin In Complex With An Oxazolopyridine Inhibitor 2
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2005-09-27 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 501 |
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-09-27
Ligands: 501
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Crystal Structure Of Human Beta Secretase Complexed With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2004-11-09 Classification: HYDROLASE Ligands: 32P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-11-09
Ligands: 32P
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Crystal Structure Of Thrombin In Complex With L-378,622
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2004-04-06 Classification: BLOOD CLOTTING,HYDROLASE/INHIBITOR Ligands: CDA |
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-04-06
Ligands: CDA
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Thrombin-Hirugen_L-378,650
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2004-04-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CDB |
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-04-06
Ligands: CDB
