Search Count: 16
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Structure-Guided Discovery Of Selective Usp7 Inhibitors With In Vivo Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2024-11-06 Classification: HYDROLASE Ligands: R4D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: R4D
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Structure-Guided Discovery Of Selective Usp7 Inhibitors With In Vivo Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.06 Å Release Date: 2024-11-06 Classification: HYDROLASE Ligands: A1ICU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1ICU
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Structure-Guided Discovery Of Selective Usp7 Inhibitors With In Vivo Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2024-11-06 Classification: HYDROLASE Ligands: A1ICV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1ICV
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Structure-Guided Discovery Of Selective Usp7 Inhibitors With In Vivo Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.76 Å Release Date: 2024-11-06 Classification: HYDROLASE Ligands: A1ICS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1ICS
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Structure-Guided Discovery Of Selective Usp7 Inhibitors With In Vivo Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2024-11-06 Classification: HYDROLASE Ligands: A1ICW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1ICW
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Structure-Guided Discovery Of Selective Usp7 Inhibitors With In Vivo Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2024-11-06 Classification: HYDROLASE Ligands: A1ICT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1ICT
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Structure-Guided Discovery Of Selective Usp7 Inhibitors With In Vivo Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.37 Å Release Date: 2024-11-06 Classification: HYDROLASE Ligands: A1ICX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1ICX
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Structure-Guided Discovery Of Selective Usp7 Inhibitors With In Vivo Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2024-11-06 Classification: HYDROLASE Ligands: A1ICO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1ICO
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Structure Of Mcl-1 Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2021-10-13 Classification: APOPTOSIS Ligands: U6Q, MG, PG6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: U6Q, MG, PG6
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Structure Of Mcl-1 Complex With Compound 6B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2021-10-13 Classification: APOPTOSIS Ligands: U6N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: U6N
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Structure Of Mcl-1 In Complex With Compound 2G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2020-11-18 Classification: APOPTOSIS Ligands: OJT, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: OJT, CL
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Structure Of Mbp-Mcl-1 In Complex With Compound 3E
Organism: Escherichia coli o157:h7, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2020-11-18 Classification: APOPTOSIS Ligands: CL, OJW |
Organism: Escherichia coli o157:h7, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: CL, OJW
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Structure Of Mbp-Mcl-1 In Complex With Compound 4D
Organism: Escherichia coli o157:h7, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-11-18 Classification: APOPTOSIS Ligands: CL, OK2 |
Organism: Escherichia coli o157:h7, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: CL, OK2
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Structure Of Mbp-Mcl-1 In Complex With Compound 9M
Organism: Escherichia coli o157:h7, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2020-11-18 Classification: APOPTOSIS Ligands: OK5 |
Organism: Escherichia coli o157:h7, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: OK5
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Crystal Structure Of Bcl-2 In Complex With The Novel Orally Active Inhibitor S55746
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2018-11-07 Classification: APOPTOSIS Ligands: F3Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-07
Ligands: F3Q
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Crystal Structure Of The Mbp-Mcl1 Complex With Highly Selective And Potent Inhibitor Of Mcl1
Organism: Escherichia coli o157:h7, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-10-26 Classification: APOPTOSIS/INHIBITOR Ligands: 70R |
Organism: Escherichia coli o157:h7, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-26
Ligands: 70R
