Search Count: 13
![]() |
Estrogen Receptor Mutant L536S
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: L5B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: L5B
![]() |
Discovery And Optimization Of Pyrimidone Indoline Amide Pi3Kbeta Inhibitors For The Treatment Of Phosphatase And Tensin Homologue (Pten)-Deficient Cancers
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-01-15 Classification: TRANSFERASE Ligands: J82 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2014-01-15
Ligands: J82
![]() |
X-Ray Structure Of Pi3K-Gamma Bound To A 4-(Morpholin-4-Yl)- (6-Oxo-1,6-Dihydropyrimidin-2-Yl)Amide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2012-11-14 Classification: Transferase/Transferase Inhibitor Ligands: 0W7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: 0W7
![]() |
Discovery And Optimization Of New Benzimidazole- And Benzoxazole-Pyrimidone Selective Pi3Kbeta Inhibitors For The Treatment Of Phosphatase And Tensin Homologue (Pten)-Deficient Cancers
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2012-05-16 Classification: TRANSFERASE Ligands: VWN |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: VWN
![]() |
Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2011-10-26 Classification: CHAPERONE Ligands: YK9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: YK9
![]() |
Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YJW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YJW
![]() |
Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YJX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YJX
![]() |
Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YJW, YJX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YJW, YJX
![]() |
Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YKB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YKB
![]() |
Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YKC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YKC
![]() |
Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YKE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YKE
![]() |
Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YKI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YKI
![]() |
Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YKJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YKJ
