Search Count: 7
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Bivalent Binding To Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2016-09-28 Classification: TRANSCRIPTION Ligands: ETU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-28
Ligands: ETU
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Bivalent Binding To Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2016-09-28 Classification: TRANSCRIPTION Ligands: K6K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-28
Ligands: K6K
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The First Bet Bromodomain Of Brd4 Bound To Compound 13 In A Bivalent Manner
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2016-09-21 Classification: Transcription Factor Ligands: XNH, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: XNH, GOL
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A Novel Oral Selective Estrogen Receptor Down-Regulator, Azd9496, Drives Tumour Growth Inhibition In Estrogen Receptor Positive And Esr1 Mutant Models
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2015-12-16 Classification: SIGNALING PROTEIN Ligands: KE9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: KE9
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Optimization Of A Novel Binding Motif To To (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-Fluoro-2-Methylpropyl)-3-Methyl-2,3,4,9-Tetrahydro-1H- Pyrido(3,4-B)Indol-1-Yl)Phenyl)Acrylic Acid (Azd9496), A Potent And Orally Bioavailable Selective Estrogen Receptor Downregulator And Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-10-14 Classification: SIGNALING PROTEIN Ligands: XBR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: XBR
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Optimization Of A Novel Binding Motif To To (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-Fluoro-2-Methylpropyl)-3-Methyl-2,3,4,9-Tetrahydro-1H- Pyrido(3,4-B)Indol-1-Yl)Phenyl)Acrylic Acid (Azd9496), A Potent And Orally Bioavailable Selective Estrogen Receptor Downregulator And Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-10-14 Classification: SIGNALING PROTEIN Ligands: GW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: GW5
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Oxyphenylpropenoic Acids As Oral Selective Estrogen Receptor Down- Regulators.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2015-04-22 Classification: SIGNALING PROTEIN Ligands: 85Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: 85Z