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Search Count: 25

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8BJU image
Human Wee1 Kinase In Complex With Inhibitor 1-[6-(1-Hydroxy-1-Methyl-Ethyl)-Pyridin-2-Yl]-2-(2-Methoxy-Phenyl)-6-[4-(4-Methyl-Piperazin-1-Yl)-Phenylamino]-1,2-Dihydro-Pyrazolo[3,4-D]Pyrimidin-3-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.53 Å Release Date: 2023-05-31
Classification: TRANSFERASE
Ligands: QT9

8BJT image
Structure Of Human Plk1 In Complex With 2-Allyl-1-[6-(1-Hydroxy-1-Methyl-Ethyl)-Pyridin-2-Yl]-6-[4-(4-Methyl-Piperazin-1-Yl)-Phenylamino]-1,2-Dihydro-Pyrazolo[3,4-D]Pyrimidin-3-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.19 Å Release Date: 2023-04-26
Classification: TRANSFERASE
Ligands: ACT, 8X7, ZN

7R60 image
Btk In Complex With 18A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.94 Å Release Date: 2021-10-06
Classification: TRANSFERASE/INHIBITOR
Ligands: 2IE

7R61 image
Btk In Complex With 25A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.52 Å Release Date: 2021-10-06
Classification: TRANSFERASE/INHIBITOR
Ligands: 2IJ, DMS

7KXL image
Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.84 Å Release Date: 2021-05-19
Classification: TRANSFERASE
Ligands: X9J, DMS

7KXM image
Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.33 Å Release Date: 2021-05-19
Classification: TRANSFERASE
Ligands: X9M

7KXN image
Btk1 Soaked With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.34 Å Release Date: 2021-05-19
Classification: TRANSFERASE
Ligands: X9P, DMS

7KXO image
Btk1 Soaked With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.94 Å Release Date: 2021-05-19
Classification: TRANSFERASE
Ligands: X9S, DMS

7KXP image
Btk1 Soaked With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.83 Å Release Date: 2021-05-19
Classification: TRANSFERASE
Ligands: X9V, DMS

7KXQ image
Btk1 Soaked With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.38 Å Release Date: 2021-05-19
Classification: TRANSFERASE
Ligands: DMS, X9Y

6OMU image
Structure Of Human Bruton'S Tyrosine Kinase In Complex With Evobrutinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.41 Å Release Date: 2019-08-14
Classification: Transferase/Transferase Inhibitor
Ligands: CL, MZJ

6N9P image
Discovery Of Affinity-Based Probes For Btk Occupancy Assay
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.23 Å Release Date: 2019-02-06
Classification: IMMUNE SYSTEM
Ligands: KHD

6DI0 image
Crystal Structure Of Btk In Complex With Fragment Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.30 Å Release Date: 2018-10-17
Classification: TRANSFERASE/TRANSFERASE Inhibitor
Ligands: GJG

6DI1 image
Crystal Structure Of Btk In Complex With Covalent Fragment Ligand
Organism: homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.10 Å Release Date: 2018-10-17
Classification: TRANSFERASE/TRANSFERASE inhibitor
Ligands: GJD

6DI3 image
Crystal Structure Of Btk In Complex With Fragment Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2018-09-05
Classification: TRANSFERASE/TRANSFERASE Inhibitor
Ligands: GJA

6DI5 image
Crystal Structure Of Btk In Complex With Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.42 Å Release Date: 2018-09-05
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: GJ7, DMS

6DI9 image
Crystal Structure Of Btk In Complex With Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.25 Å Release Date: 2018-09-05
Classification: TRANSFERASE/TRANSFERASE Inhibitor
Ligands: GJJ, DMS

4ZZH image
Sirt1/Activator Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.10 Å Release Date: 2015-07-15
Classification: Hydrolase/hydrolase activator
Ligands: ZN, 4TO

4ZZI image
Sirt1/Activator/Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.73 Å Release Date: 2015-07-15
Classification: Hydrolase/hydrolase inhibitor
Ligands: 4TQ, 1NS, ZN

4ZZJ image
Sirt1/Activator/Substrate Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.74 Å Release Date: 2015-07-15
Classification: HYDROLASE
Ligands: ZN, CNA, 4TQ, GOL
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