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Tricyclic Indazoles A Novel Class Of Selective Estrogen Receptor Degrader Antagonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2019-01-23 Classification: DNA BINDING PROTEIN Ligands: H8W |
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A Novel Oral Selective Estrogen Receptor Down-Regulator, Azd9496, Drives Tumour Growth Inhibition In Estrogen Receptor Positive And Esr1 Mutant Models
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2015-12-16 Classification: SIGNALING PROTEIN Ligands: KE9 |
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Optimization Of A Novel Binding Motif To To (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-Fluoro-2-Methylpropyl)-3-Methyl-2,3,4,9-Tetrahydro-1H- Pyrido(3,4-B)Indol-1-Yl)Phenyl)Acrylic Acid (Azd9496), A Potent And Orally Bioavailable Selective Estrogen Receptor Downregulator And Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-10-14 Classification: SIGNALING PROTEIN Ligands: XBR |
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Optimization Of A Novel Binding Motif To To (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-Fluoro-2-Methylpropyl)-3-Methyl-2,3,4,9-Tetrahydro-1H- Pyrido(3,4-B)Indol-1-Yl)Phenyl)Acrylic Acid (Azd9496), A Potent And Orally Bioavailable Selective Estrogen Receptor Downregulator And Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-10-14 Classification: SIGNALING PROTEIN Ligands: GW5 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2013-02-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0XZ, GOL |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2010-10-27 Classification: TRANSPORT PROTEIN Ligands: IMX |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2010-10-27 Classification: TRANSPORT PROTEIN Ligands: IPX, PO4 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2010-10-27 Classification: TRANSPORT PROTEIN Ligands: IQX |
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Structure Of The Tie2 Kinase Domain In Complex With A Thiazolopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2009-11-03 Classification: TRANSFERASE Ligands: QQ1 |