Search Count: 35
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Crystal Structure Of Human Naa50 In Complex With A Cofactor Derived Inhibitor (Compound 1)
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: COA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: COA
 |
Crystal Structure Of Human Naa50 In Complex With A Truncated Cofactor Derived Inhibitor (Compound 2)
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: U44 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: U44
 |
Crystal Structure Of Human Naa50 In Complex With An Inhibitor (Compound 3) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: COA, U3V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: COA, U3V
 |
Crystal Structure Of Human Naa50 In Complex With Coa And An Inhibitor (Compound 4A) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2020-07-01 Classification: TRANSFERASE Ligands: COA, U2J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: COA, U2J
 |
Crystal Structure Of Human Naa50 In Complex With Accoa And An Inhibitor (Compound 4A) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.07 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: ACO, U2J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: ACO, U2J
 |
Crystal Structure Of Human Naa50 In Complex With Accoa And An Inhibitor (Compound 4B) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: ACO, U3Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: ACO, U3Y
 |
Structure Of Human Anaplastic Lymphoma Kinase In Complex With 2-[(1R)-1-{[2-Amino-5-(1,3-Dimethyl-1H-Pyrazol-4-Yl)Pyridin-3-Yl]Oxy}Ethyl]-4-Fluoro-N,N-Dimethylbenzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2016-08-17 Classification: Transferase/Transferase Inhibitor Ligands: 6YL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-17
Ligands: 6YL
 |
Structure Of C1156Y Mutant Human Anaplastic Lymphoma Kinase In Complex With Pf-06463922 ((10R)-7-Amino-12-Fluoro-2,10,16-Trimethyl- 15-Oxo-10,15,16,17-Tetrahydro-2H-8,4-(Metheno)Pyrazolo(4,3-H)(2,5,11) Benzoxadiazacyclotetradecine-3-Carbonitrile).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: 5P8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: 5P8
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Structure Of C1156Y,L1198F Mutant Human Anaplastic Lymphoma Kinase In Complex With Pf-06463922 ((10R)-7-Amino-12-Fluoro-2,10,16-Trimethyl- 15-Oxo-10,15,16,17-Tetrahydro-2H-8,4-(Metheno)Pyrazolo(4,3-H)(2,5,11) Benzoxadiazacyclotetradecine-3-Carbonitrile).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: 5P8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: 5P8
 |
Structure Of L1198F Mutant Human Anaplastic Lymphoma Kinase In Complex With Pf-06463922 ((10R)-7-Amino-12-Fluoro-2,10,16-Trimethyl- 15-Oxo-10,15,16,17-Tetrahydro-2H-8,4-(Metheno)Pyrazolo(4,3-H)(2,5,11) Benzoxadiazacyclotetradecine-3-Carbonitrile).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: 5P8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: 5P8
 |
Structure Of L1198F Mutant Human Anaplastic Lymphoma Kinase In Complex With Crizotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: VGH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: VGH
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Structure Of C1156Y,L1198F Mutant Human Anaplastic Lymphoma Kinase In Complex With Crizotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: VGH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: VGH
 |
Structure Of C1156Y Mutant Human Anaplastic Lymphoma Kinase In Complex With Crizotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: VGH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: VGH
 |
Structure Of The Human Anaplastic Lymphoma Kinase In Complex With Pf- 06463922 ((10R)-7-Amino-12-Fluoro-2,10,16-Trimethyl-15-Oxo-10,15,16, 17-Tetrahydro-2H-8,4-(Metheno)Pyrazolo(4,3-H)(2,5,11) Benzoxadiazacyclotetradecine-3-Carbonitrile).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2014-05-28 Classification: TRANSFERASE Ligands: 5P8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-28
Ligands: 5P8
 |
Structure Of L1196M Mutant Human Anaplastic Lymphoma Kinase In Complex With Pf-06463922 ((10R)-7-Amino-12-Fluoro-2,10,16-Trimethyl- 15-Oxo-10,15,16,17-Tetrahydro-2H-8,4-(Metheno)Pyrazolo(4,3-H)(2,5,11) Benzoxadiazacyclotetradecine-3-Carbonitrile).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2014-05-28 Classification: TRANSFERASE Ligands: 5P8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-28
Ligands: 5P8
 |
Structure Of The Human Anaplastic Lymphoma Kinase In Complex With The Inhibitor 2-((1R)-1-((3-Amino-6-(2-Methoxypyridin-3-Yl)Pyrazin-2-Yl) Oxy)Ethyl)-4-Fluoro-N-Methylbenzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2014-05-28 Classification: TRANSFERASE Ligands: YPW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-28
Ligands: YPW
 |
Structure Of The Human Anaplastic Lymphoma Kinase In Complex With The Inhibitor 3-((1R)-1-(5-Fluoro-2-(2H-1,2,3-Triazol-2-Yl)Phenyl)Ethoxy)- 5-(3-(Methylsulfonyl)Phenyl)Pyridin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2014-05-28 Classification: TRANSFERASE Ligands: GWH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-28
Ligands: GWH
 |
Structure Of The Human Anaplastic Lymphoma Kinase In Complex With The Inhibitor (10R)-7-Amino-12-Fluoro-1,3,10,16-Tetramethyl-16,17-Dihydro- 1H-8,4-(Metheno)Pyrazolo(4,3-H)(2,5,11)Benzoxadiazacyclotetradecin-15(10H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-05-28 Classification: TRANSFERASE Ligands: IV7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-28
Ligands: IV7
 |
Structure Of The Human Anaplastic Lymphoma Kinase In Complex With The Inhibitor 3-((1R)-1-(5-Fluoro-2-Methoxyphenyl)Ethoxy)-5-(1-Methyl-1H- 1,2,3-Triazol-5-Yl)Pyridin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2014-05-28 Classification: TRANSFERASE Ligands: 3U9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-28
Ligands: 3U9
 |
Structure Of The Human Anaplastic Lymphoma Kinase In Complex With The Inhibitor (5R)-8-Amino-3-Fluoro-5,19-Dimethyl-20-Oxo-5,18,19,20- Tetrahydro-7,11-(Azeno)Pyrido(2',1':2,3)Imidazo(4,5-H)(2,5,11) Benzoxadiazacyclotetradecine-14-Carbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2014-05-28 Classification: TRANSFERASE Ligands: KVC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-28
Ligands: KVC