Search Count: 93
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Cryo-Em Structure Of Ccr6 Bound By Pf-07054894 And Oxm2
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY Resolution:3.35 Å Release Date: 2025-10-01 Classification: MEMBRANE PROTEIN Ligands: A1A1W, A1CH1 |
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY
Release Date: 2025-10-01
Ligands: A1A1W, A1CH1
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Pad2 With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2025-07-30 Classification: HYDROLASE Ligands: A1CE0, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-30
Ligands: A1CE0, CA
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Structure Of The Type Ii Thioesterase Borb From The Borrelidin Biosynthetic Cluster
Organism: Streptomyces sp. wac02707
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2020-05-06 Classification: BIOSYNTHETIC PROTEIN |
Organism: Streptomyces sp. wac02707
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
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Crystal Structure Of Tyk2 Kinase With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2020-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: R5D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R5D
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Crystal Structure Of Tyk2 Kinase With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: R4Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R4Y
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Crystal Structure Of Tyk2 Kinase With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2020-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: R4V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R4V
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Crystal Structure Of Tyk2 Kinase With Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: R4S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R4S
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Crystal Structure Of Jak1 Kinase With Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2020-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: R4S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R4S
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A Secreted Lysm Effector Of The Wheat Pathogen Zymoseptoria Tritici Protects The Fungal Hyphae Against Chitinase Hydrolysis Through Ligand-Dependent Polymerisation Of Lysm Homodimers
Organism: Zymoseptoria tritici ipo323
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2019-10-16 Classification: HYDROLASE Ligands: CL |
Organism: Zymoseptoria tritici ipo323
Method: X-RAY DIFFRACTION
Release Date: 2019-10-16
Ligands: CL
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Tyk2 With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: G5D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: G5D
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Tyk2 With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: G4J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: G4J
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Jak1 With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: G4J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: G4J
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Crystal Structure Of Itk In Complex With Compound 1 [4-(Carbamoylamino)-1-(Naphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M0Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: M0Y
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Crystal Structure Of Itk In Complex With Compound 5 {4-(Carbamoylamino)-1-(7-Methoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide}
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M0Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: M0Z
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Crystal Structure Of Itk In Complex With Compound 7 [4-(Carbamoylamino)-1-(7-Ethoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 1YZ
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Crystal Structure Of Itk In Complex With Compound 8 [4-(Carbamoylamino)-1-(7-Propoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1E0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 1E0
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Crystal Structure Of Itk In Complex With Compound 9 [4-(Carbamoylamino)-1-[7-(Propan-2-Yloxy)Naphthalen-1-Yl]-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QWS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: QWS
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Crystal Structure Of Itk In Complex With Compound 9 [4-(Carbamoylamino)-1-[7-(Propan-2-Yloxy)Naphthalen-1-Yl]-1H-Pyrazole-3-Carboxamide] And Adp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QWS, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: QWS, ADP
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Cladosporium Fulvum Lysm Effector Ecp6 In Complex With A Beta-1,4- Linked N-Acetyl-D-Glucosamine Tetramer
Organism: Passalora fulva
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2013-07-17 Classification: SUGAR BINDING PROTEIN Ligands: NAG |
Organism: Passalora fulva
Method: X-RAY DIFFRACTION
Release Date: 2013-07-17
Ligands: NAG
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Cladosporium Fulvum Lysm Effector Ecp6 In Complex With A Beta-1,4- Linked N-Acetyl-D-Glucosamine Tetramer: I3C Heavy Atom Derivative
Organism: Passalora fulva
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-07-17 Classification: SUGAR BINDING PROTEIN Ligands: NAG, I3C |
Organism: Passalora fulva
Method: X-RAY DIFFRACTION
Release Date: 2013-07-17
Ligands: NAG, I3C
