Structural Entry Filters:

Search Count: 30

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8C6P image
Fragment Screening Hit I Bound To Endothiapepsin

8C6Q image
Fragment Screening Hit Ii Bound To Endothiapepsin

8C6S image
Fragment Screening Hit Iii Bound To Endothiapepsin

8C6T image
Fragment Screening Hit Iv Bound To Endothiapepsin

8C70 image
Pyrrolidine Fragment 1 Bound To Endothiapepsin

8C71 image
Pyrrolidine Fragment 5B Bound To Endothiapepsin

8C72 image
Pyrrolidine Fragment 10B Bound To Endothiapepsin

8C74 image
Pyrrolidine Fragment 10D Bound To Endothiapepsin

7OVI image
Protein Kinase Mkk7 In Complex With Phenethyltriazole-Substituted Pyrazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2022-07-20
Classification: TRANSFERASE
Ligands: 2GI

7OVJ image
Protein Kinase Mkk7 In Complex With Difluoro-Phenethyltriazole-Substituted Pyrazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2022-07-20
Classification: TRANSFERASE
Ligands: 24N

7OVK image
Protein Kinase Mkk7 In Complex With 5-Bromo-2-Hydroxyphenyl-Substituted Pyrazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.05 Å Release Date: 2022-07-20
Classification: TRANSFERASE
Ligands: GOL, 2I5

7OVL image
Protein Kinase Mkk7 In Complex With Methoxycyclohexyl-Substituted Indazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.90 Å Release Date: 2022-07-20
Classification: TRANSFERASE
Ligands: 1XZ

7OVM image
Protein Kinase Mkk7 In Complex With Cyclobutyl-Substituted Indazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.90 Å Release Date: 2022-07-20
Classification: TRANSFERASE
Ligands: 21I

7OVN image
Protein Kinase Mkk7 In Complex With Tolyl-Substituted Indazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.90 Å Release Date: 2022-07-20
Classification: TRANSFERASE
Ligands: 2I8

5OMG image
P38Alpha In Complex With Pyrazolobenzothiazine Inhibitor Coxp4M12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2019-03-13
Classification: TRANSFERASE
Ligands: BOG, 9Y8

5OMH image
P38Alpha In Complex With Pyrazolobenzothiazine Inhibitor Coxh11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 2019-03-13
Classification: TRANSFERASE
Ligands: 9Y5

5N63 image
Crystal Structure Of P38Alpha In Complex With Lipid Pocket Ligand 9C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2017-09-20
Classification: TRANSFERASE
Ligands: 8OW

5N64 image
Crystal Structure Of P38Alpha In Complex With Lipid Pocket Ligand 9G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2017-09-20
Classification: TRANSFERASE
Ligands: 8OH

5N65 image
Crystal Structure Of P38Alpha In Complex With Lipid Pocket Ligand 9H
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2017-09-20
Classification: TRANSFERASE
Ligands: 8OT

5N66 image
Crystal Structure Of P38Alpha In Complex With Lipid Pocket Ligand 9J
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2017-09-20
Classification: TRANSFERASE
Ligands: BW1, B96
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